Search Count: 19
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Crystal Structure Of Menin In Complex With Inhibitor Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVE
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Crystal Structure Of Menin In Complex With Inhibitor Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVF, K, EPE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVF, K, EPE, SO4
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Crystal Structure Of Menin In Complex With Inhibitor Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-01-15 Classification: PROTEIN BINDING/INHIBITOR Ligands: A1AVG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-15
Ligands: A1AVG
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Tas-120 Covalent Structure With Fgfr2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2025-01-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1AFR, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: A1AFR, GOL, SO4
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Tas-120 Covalent Structure With Fgfr2 Molecular Brake Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2025-01-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TZ0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: TZ0, SO4
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Tas-120 Covalent Structure With Fgfr2 Molecular Brake Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2025-01-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TZ0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: TZ0, SO4
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Tas-120 Covalent Structure With Fgfr2 Molecular Brake Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2025-01-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TZ0, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: TZ0, GOL, SO4
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Kras G12D In Complex With Mrtx-1133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2021-12-22 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GDP, 6IC, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: GDP, 6IC, MG
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Crystal Structure Of Kras G12D With Compound 15 (4-(4-[(1R,5S)-3,8-Diazabicyclo[3.2.1]Octan-3-Yl]-8-Fluoro-2-{[(2S)-1-Methylpyrrolidin-2-Yl]Methoxy}Pyrido[4,3-D]Pyrimidin-7-Yl)Naphthalen-2-Ol) Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2021-12-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, 7L8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: GDP, MG, 7L8
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Crystal Structure Of Kras G12D With Compound 25 (4-(4-[(1R,5S)-3,8-Diazabicyclo[3.2.1]Octan-3-Yl]-8-Fluoro-2-{[(2R,4R,7As)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl]Methoxy}Pyrido[4,3-D]Pyrimidin-7-Yl)Naphthalen-2-Ol) Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2021-12-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, 7NL, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: GDP, MG, 7NL, GOL, EDO
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Crystal Structure Of Kras G12D With Compound 24 (4-(4-[(1R,5S)-3,8-Diazabicyclo[3.2.1]Octan-3-Yl]-8-Fluoro-2-{[(2S,4S,7Ar)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl]Methoxy}Pyrido[4,3-D]Pyrimidin-7-Yl)Naphthalen-2-Ol) Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2021-12-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, 7NZ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: GDP, 7NZ, MG
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Kras G12D In Complex With Compound 5B (7-(8-Chloronaphthalen-1-Yl)-8-Fluoro-2-{[(2S)-1-Methylpyrrolidin-2-Yl]Methoxy}-4-(Piperazin-1-Yl)Pyrido[4,3-D]Pyrimidine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-12-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, MG, 7IZ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: GDP, MG, 7IZ, GOL
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Crystal Structure Of Kras G12D With Compound 36 (4-[(1R,5S)-3,8-Diazabicyclo[3.2.1]Octan-3-Yl]-7-(8-Ethynyl-7-Fluoronaphthalen-1-Yl)-8-Fluoro-2-{[(4S,7As)-Tetrahydro-1H-Pyrrolizin-7A(5H)-Yl]Methoxy}Pyrido[4,3-D]Pyrimidine) Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2021-12-22 Classification: HYDROLASE/INHIBITOR Ligands: GDP, 7OE, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: GDP, 7OE, MG
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Crystal Structure Of Arl2 Gtpase-Activating Protein Tubulin Cofactor C (Tbcc)
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-08-12 Classification: CHAPERONE Ligands: SO4 |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c)
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: SO4
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Crystal Structure Of Assimilatory Adenosine 5'-Phosphosulfate Reductase With Bound Aps
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2006-09-19 Classification: OXIDOREDUCTASE Ligands: SF4, ADX |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2006-09-19
Ligands: SF4, ADX
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Structure Of A Chordin-Like Cysteine-Rich Repeat (Vwc Module) From Collagen Iia
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2004-10-05 Classification: STRUCTURAL PROTEIN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2004-10-05
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Mycobacterium Smegmatis Stf0 Sulfotransferase With Trehalose
Organism: Mycobacterium smegmatis
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2004-07-20 Classification: TRANSFERASE |
Organism: Mycobacterium smegmatis
Method: X-RAY DIFFRACTION
Release Date: 2004-07-20
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Nmr Structure Of 16Th Module Of Immune Adherence Receptor, Cr1 (Cd35)
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Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2004-05-04
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Nmr Study Of The Third Tb Domain From Latent Transforming Growth Factor-Beta Binding Protein-1
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2003-08-26 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2003-08-26
