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9TDA image
Erap1 In Complex With 1-[2-(5-Bromo-7-Fluoro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid

9TD3 image
Erap1 In Complex With 1-[2-(6-Bromo-2,2-Difluoro-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9TD4 image
Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9TD5 image
Erap1 In Complex With 1-[2-(5-Chloro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9TD7 image
Erap1 In Complex With 1-[2-(3-Oxo-6-Phenyl-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9GJN image
Erap1 In Complex With 1-[2-(3-Oxo-3,4-Dihydro-2H-1,4-Benzothiazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9GJS image
Erap1 In Complex With 1-[2-(6-Bromo-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid

9GK6 image
Erap1 In Complex With 1-[2-(6-Chloro-3-Oxo-3,4-Dihydro-2H-1,4-Benzothiazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9GKE image
Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

7PI4 image
Fak Protac Gsk215 In Complex With Fak And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.24 Å Release Date: 2021-09-29
Classification: TRANSFERASE
Ligands: 7QB, PEG, EDO, CA

6FFE image
Human Brd2 C-Terminal Bromodomain With 2-((4-Acetyl-3-Cyclopropyl-3,4-Dihydroquinoxalin-1(2H)-Yl)Methyl)Benzoic Acid

6FFF image
Human Brd2 C-Terminal Bromodomain With (S)-5-(1-Acetyl-2-Cyclopropyl-4-(2-(Hydroxymethyl)Benzyl)-1,2,3,4-Tetrahydroquinoxalin-6-Yl)Pyrimidine-2-Carboxamide

6FFG image
Human Brd2 C-Terminal Bromodomain With (S)-1-(2-Cyclopropyl-4-(2-(Hydroxymethyl)Benzyl)-6-(1,2,3,6-Tetrahydropyridin-4-Yl)-3,4-Dihydroquinoxalin-1(2H)-Yl)Ethanone

5G4R image
Bromodomain Of Human Brpf1 With N-1,3-Dimethyl-6-2R-2- Methylpiperazin-1-Yl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl-2- Methoxybenzamide

5G4S image
Bromodomain Of Human Brpf1 With N-1,3-Dimethyl-6-2R-2- Methylpiperazin-1-Yl-2-Oxo-2,3-Dihydro-1H-1,3-Benzodiazol-5-Yl-N- Ethyl-2-Methoxybenzamide
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