Search Count: 45
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C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, SO4
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 98A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 98A
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9XO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9XO
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9OO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9OO
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9VV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9VV
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: EDO, 9WU, BR, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: EDO, 9WU, BR, CL
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9KI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9KI
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C-Kit T670I Mutated Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI
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Pdgfra T674I Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, PEG
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Pdgfra T674I Mutant Kinase Domain In Complex With Avapritinib Derivative 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9OO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9OO, PEG
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Pdgfra Wild-Type Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2023-12-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
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Apo Crystal Structure Of Pdgfra-T674I Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-12-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
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Crystal Structure Of Egfr-T790M/V948R In Complex With Ldc8201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: SO4, R1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: SO4, R1W
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Crystal Structure Of Egfr-T790M/V948R In Complex With Poziotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: R2E, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: R2E, SO4, EDO
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Crystal Structure Of Egfr-T790M/V948R In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: R28, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: R28, SO4
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Crystal Structure Of Egfr-Wt In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: R28, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: R28, MES
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Crystal Structure Of Egfr-T790M/V948R In Complex With Osimertinib And Eai045
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-11-11 Classification: TRANSFERASE Ligands: Q6K, 9LL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-11
Ligands: Q6K, 9LL, SO4
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Crystal Structure Of Egfr-T790M/V948R In Complex With Mavelertinib And Eai001
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-11-11 Classification: TRANSFERASE Ligands: 8BS, SO4, 57N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-11
Ligands: 8BS, SO4, 57N
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Crystal Structure Of Egfr-T790M/V948R In Complex With Spebrutinib And Eai001
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-11-11 Classification: TRANSFERASE Ligands: 57N, 7G9, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-11
Ligands: 57N, 7G9, SO4, CL
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Crystal Structure Of Egfr T790M/V948R In Complex With Covalent Pyrrolopyrimidine 14D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-09-30 Classification: TRANSFERASE Ligands: N7K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: N7K, SO4
