Search Count: 10
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Benzodiazepine Hts Hit Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: W89, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: W89, ZN, NA
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Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Wo2020264398 Ex23)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: Z3N, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: Z3N, ZN, NA
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Crystal Structure Of The E3 Ubiquitin Ligase Cbl-B With An Allosteric Inhibitor (Benzodiazepine Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2023-11-22 Classification: LIGASE Ligands: W7R, ZN, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: W7R, ZN, NA
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Estrogen Receptor Alpha In Complex With Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2023-02-01 Classification: TRANSCRIPTION Ligands: H09 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: H09
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-02-01 Classification: GENE REGULATION Ligands: GZI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: GZI
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
