Search Count: 9
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Structure Of Sars-Cov-2 Main Protease In Complex With A Covalent Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-05-15 Classification: VIRAL PROTEIN Ligands: YDL |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-05-15
Ligands: YDL
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Aminomethyl-Derived Beta Secretase (Bace1) Inhibitors: Engaging Gly230 Without An Anilide Functionality
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2017-01-11 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: P6U, IOD, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: P6U, IOD, EDO
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Aminomethyl-Derived Beta Secretase (Bace1) Inhibitors: Engaging Gly230 Without An Anilide Functionality
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2017-01-11 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 74B, IOD, NA, GOL, DMS, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 74B, IOD, NA, GOL, DMS, CL
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Structure Of Cytochrome P450 2D6 (Cyp2D6) Bace1 Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2017-01-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: HEM, ZN, P6U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: HEM, ZN, P6U
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Structure Of Cytochrome P450 2D6 (Cyp2D6) Bace1 Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-01-11 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: HEM, ZN, P6M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: HEM, ZN, P6M
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Crystal Structure Of Gsk-3Beta Complexed With Pf-04802367, A Highly Selective Brain-Penetrant Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-09-21 Classification: TRANSFERASE Ligands: 6QH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6QH, SO4
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Crystal Structure Of Bace With Compound 14G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2012-10-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0UP, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: 0UP, ZN
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Crystal Structure Of Bace With Compound 12A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-10-03 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 0UQ, ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: 0UQ, ZN, EDO
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6-Amino-4-(Pyrimidin-4-Yl)Pyridones: Novel Glycogen Synthase Kinase-3 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-06-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 55E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: 55E
