Search Count: 22
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Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: EDO
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C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: B49, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: B49, EDO, CL
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C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: XIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: XIN
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C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: STI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: STI, CL
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C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 0LI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 0LI, CL
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C-Kit Kinase Domain In Complex With S116836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: A1H4U, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1H4U, CL
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C-Kit Kinase Domain In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: STU
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C-Kit Kinase Domain In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 6T2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 6T2
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C-Kit Kinase Domain In Complex With Idrx-42 Via Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: K3R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: K3R, CL
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Crystal Structure Of Egfr-T790M/V948R In Complex With Ldc8201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: SO4, R1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: SO4, R1W
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Crystal Structure Of Egfr-T790M/V948R In Complex With Poziotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: R2E, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: R2E, SO4, EDO
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Crystal Structure Of Egfr-T790M/V948R In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: R28, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: R28, SO4
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Crystal Structure Of Egfr-Wt In Complex With Tak-788
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-02-23 Classification: TRANSFERASE Ligands: R28, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: R28, MES
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Co-Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-09-08 Classification: TRANSFERASE Ligands: UCE, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: UCE, ACT
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Co-Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-09-08 Classification: TRANSFERASE Ligands: ACT, UC8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ACT, UC8
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 16A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-10-16 Classification: TRANSFERASE Ligands: L1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: L1Z
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 15C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-10-16 Classification: TRANSFERASE Ligands: L1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: L1W
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor Borussertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-03-20 Classification: TRANSFERASE Ligands: G4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: G4K
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4T
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4Q
