Search Count: 17
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Human Pxr Lbd Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: 07F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: 07F
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Human Pxr Lbd Bound To Gsk003
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: 5YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: 5YX
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Human Pxr Lbd Bound To Gsk002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: 5YU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: 5YU
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Human Pxr Lbd Bound To Gsk001
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-25 Classification: GENE REGULATION Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-25
Ligands: P06
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Rip2 Kinase Catalytic Domain Complex With 5Amino1Tertbutyl3(3Methoxyphenyl)1H Pyrazole4Carboxamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: M5W, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: M5W, CA
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Rip2 Kinase Catalytic Domain Complex With (5S,6S,8R)-2-(Benzo[D]Thiazol-5-Yl)-6-Hydroxy-4,5,6,7,8,9-Hexahydro-5,8-Methanopyrazolo[1,5-A][1,3]Diazocine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2019-12-04 Classification: TRANSFERASE Ligands: Q9J, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-04
Ligands: Q9J, CA
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Rip2 Kinase Catalytic Domain Complex With 5-Amino-1-Phenylpyrazole-4-Carboxamide.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2019-10-23 Classification: TRANSFERASE Ligands: M2B, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: M2B, CA
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: J6H |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: J6H
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: DMS, J6N |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: DMS, J6N
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: SO4, J6Q |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: SO4, J6Q
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: SO4, CL, J6K |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: SO4, CL, J6K
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: CL, J8H |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: CL, J8H
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Rip2 Kinase Catalytic Domain Complex With N(4,5Dimethyl1Hpyrazol3Yl)7Methoxy6(2Methylpropane2Sulfonyl)Quinolin4Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-11-07 Classification: TRANSFERASE Ligands: GEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-07
Ligands: GEZ
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Compound 3 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GE, SO4
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Gsk583 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GD
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Crystal Structure Of Rip1 Kinase With A Benzo[B][1,4]Oxazepin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 65U
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Structure Of The B-Raf Kinase Domain Bound To Sb-590885
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2006-12-12 Classification: TRANSFERASE Ligands: 215 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
Ligands: 215