Search Count: 16
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Crystal Structure Of 2-(3-Alkoxy-1-Azetidinyl) Quinolines As Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: SO4, GOL, 35E, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, GOL, 35E, ZN
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2-(3-Alkoxy-1-Azetidinyl) Quinolines As Novel Pde10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2014-12-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, GOL, 35D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: ZN, SO4, GOL, 35D
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Human Gkrp Bound To Amg-2526 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-08 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TE, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 2TE, S6P, IOD, GOL, SO4
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Crystal Structure Of Pde10A With 1H-Benzimidazol-2-Yl(4-((3-(Tetrahydro-2H-Pyran-4-Yl)-2-Pyridinyl)Oxy)Phenyl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-08-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, 2W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: ZN, SO4, 2W1
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Human Gkrp Bound To Amg-0771 And Sorbitol-6-Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TF, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TF, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-2668
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TG, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TG, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-3227 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-07-30 Classification: CARBOHYDRATE BINDING PROTEIN/INHIBITOR Ligands: 2TJ, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: 2TJ, S6P, IOD, GOL, SO4
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Human Gkrp Complexed To Amg-3969 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG9, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG9, S6P, IOD, GOL, SO4
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Human Gkrp Bound To Amg-5980 And S6P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-05-07 Classification: Transferase Inhibitor Ligands: MG0, S6P, IOD, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-07
Ligands: MG0, S6P, IOD, GOL, SO4
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Crystal Structure Of Pde10A With Novel Keto-Benzimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2013-10-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, GOL, 2F4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-23
Ligands: ZN, SO4, GOL, 2F4
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Crystal Structure Of Pde10A With Novel Keto-Benzimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-10-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, 2F5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-23
Ligands: ZN, SO4, 2F5
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Pde10A Crystal Structure Complexed With Novel Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2012-03-21 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, SO4, 0JQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: ZN, SO4, 0JQ
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Benzisoxazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2008-09-09 Classification: TRANSFERASE Ligands: A96 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-09-09
Ligands: A96
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Pyridone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-06-17 Classification: TRANSFERASE Ligands: C19 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: C19
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Bisamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2008-06-17 Classification: TRANSFERASE Ligands: C92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: C92
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Pyridone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-06-17 Classification: TRANSFERASE Ligands: C52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: C52
