Search Count: 18
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
 |
Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
 |
Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
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Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
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C-Src In Complex With Atp-Chf
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-02-07 Classification: TRANSFERASE Ligands: 8BU, MG |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: 8BU, MG
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C-Src In Complex With Atp-Chcl
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: 8C6, MG, GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: 8C6, MG, GOL
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Kinase Domain Of Human Ephb1 Bound To A Quinazoline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: 7O3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: 7O3, SO4
 |
Kinase Domain Of Human Ephb1, G703C Mutant, Covalently Bound To A Quinazoline-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-05-17 Classification: TRANSFERASE Ligands: 7O3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-17
Ligands: 7O3, SO4
 |
Ephb3 Kinase Domain Covalently Bound To An Irreversible Inhibitor (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-08-10 Classification: TRANSFERASE Ligands: 6P6, DIO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 6P6, DIO
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Ephb3 Kinase Domain Covalently Bound To An Irreversible Inhibitor (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2016-08-10 Classification: TRANSFERASE Ligands: 6P8, DIO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: 6P8, DIO
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Crystal Structure Of Human Cdk8-Cyclin C In Complex With Cortistatin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-09-23 Classification: TRANSFERASE Ligands: C1I, FMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-23
Ligands: C1I, FMT
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Crystal Structure Of Kpt251 In Complex With Crm1-Ran-Ranbp1
Organism: Homo sapiens, Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-09-05 Classification: PROTEIN TRANSPORT/INHIBITOR Ligands: GNP, MG, EDO, CL, 51K, GOL |
Organism: Homo sapiens, Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: GNP, MG, EDO, CL, 51K, GOL
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Discovery Of A Small Molecule Type Ii Inhibitor Of Wild-Type And Gatekeeper Mutants Of Bcr-Abl, Pdgfralpha, Kit, And Src Kinases
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-02-15 Classification: TRANSFERASE Ligands: NG7, MES, GOL |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2012-02-15
Ligands: NG7, MES, GOL
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jq1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2010-10-06 Classification: CELL CYCLE Ligands: JQ1, IOD, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: JQ1, IOD, EDO, DMS
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Crystal Structure Of The Second Bromodomain Of Human Brd2 In Complex With The Inhibitor Jq1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2010-10-06 Classification: CELL CYCLE Ligands: JQ1, NI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: JQ1, NI, EDO
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Human Abl Kinase In Complex With Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2008-04-22 Classification: TRANSFERASE Ligands: NIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NIL
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Solution Structure Of The Cited2 Transactivation Domain In Complex With The P300 Ch1 Domain
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2003-07-01 Classification: TRANSCRIPTION/TRANSFERASE Ligands: ZN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2003-07-01
Ligands: ZN
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Nmr Structures Of The Hif-1Alpha Ctad/P300 Ch1 Complex
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2002-04-24 Classification: TRANSCRIPTION Ligands: ZN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2002-04-24
Ligands: ZN