Search Count: 28
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 20)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, WB4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, PEG, WB4
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Structure Of Human Hdac2 In Complex With An Aryl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2020-07-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, V1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: ZN, CA, SO4, PEG, V1D
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Co-Structure Of Btk Kinase Domain With L-005085737 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULV, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULV, 5WE
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Co-Structure Of Btk Kinase Domain With L-005191930 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULY, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULY, 5WE
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Co-Structure Of Btk Kinase Domain With L-005298385 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: UM4, EDO, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: UM4, EDO, BTB
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Btk-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-03-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5WH, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-23
Ligands: 5WH, 5WE
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Btk Kinase Domain With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-03 Classification: TRANSFERASE Ligands: 5WF, 5WE, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 5WF, 5WE, CL, EDO
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Discovery Of An Irreversible Hcv Ns5B Polymerase Inhibitor
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2F3, PO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: 2F3, PO4
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Hcv Ns5B Polymerase Complexed With Pyridonylindole Compound
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2013-10-09 Classification: TRANSFERASE Ligands: 8Y6, PO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: 8Y6, PO4
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Sar Development And Discovery Of Potent Indole-Based Inhibitors Of The Hepatitis C Virus Ns5B Polymerase
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: HI4, PO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: HI4, PO4
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Sar Development And Discovery Of Potent Indole-Based Inhibitors Of The Hepatitis C Virus Ns5B Polymerase
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, HI3 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: PO4, HI3
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Synthesis Of Novel 4,5-Dihydrofurano Indoles And Their Evaluation As Hcv Ns5B Polymerase Inhibitors
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, 0C1 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: PO4, 0C1
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Synthesis Of Novel 4,5-Dihydrofurano Indoles And Their Evaluation As Hcv Ns5B Polymerase Inhibitors
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-01-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, 0C2 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: PO4, 0C2
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Novel Hcv Ns5B Polymerase Inhibitors: Discovery Of Indole C2 Acyl Sulfonamides
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2011-12-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 08E, PO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: 08E, PO4
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Novel Hcv Ns5B Polymerase Inhibitors: Discovery Of Indole C2 Acyl Sulfonamides
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 08F |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2011-12-07
Ligands: 08F
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I. Novel Hcv Ns5B Polymerase Inhibitors: Discovery Of Indole 2- Carboxylic Acids With C3-Heterocycles
Organism: Hepatitis c virus isolate hc-j4
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2011-08-31 Classification: transferase/transferase INHIBITOR Ligands: PO4, 053 |
Organism: Hepatitis c virus isolate hc-j4
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PO4, 053
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I. Novel Hcv Ns5B Polymerase Inhibitors: Discovery Of Indole 2- Carboxylic Acids With C3-Heterocycles
Organism: Hepatitis c virus isolate hc-j4
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2011-08-31 Classification: transferase/transferase INHIBITOR Ligands: PO4, 054 |
Organism: Hepatitis c virus isolate hc-j4
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: PO4, 054
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I. Novel Hcv Ns5B Polymerase Inhibitors: Discovery Of Indole 2- Carboxylic Acids With C3-Heterocycles
Organism: Hepatitis c virus isolate hc-j4
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-08-31 Classification: transferase/transferase INHIBITOR Ligands: 058 |
Organism: Hepatitis c virus isolate hc-j4
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: 058
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Crystal Structure Of Catalytic Domain Of Tace With 2-(2-Aminothiazol-4-Yl)Pyrrolidine-Based Tartrate Diamides
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2011-04-20 Classification: hydrolase/hydrolase inhibitor Ligands: IPA, INN, ZN, CA, 786 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-20
Ligands: IPA, INN, ZN, CA, 786