Search Count: 40
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor Containing A Spiro-Bicyclic Group (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-08-11 Classification: HYDROLASE Ligands: ZN, SO4, CA, PEG, VJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: ZN, SO4, CA, PEG, VJV
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Structure Of Hdac2 In Complex With A Macrocyclic Inhibitor (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZLV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZLV
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Structure Of Hdac2 In Complex With An Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, V1P
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Structure Of Hdac2 In Complex With An Inhibitor (Compound 14)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZLS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZLS
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Structure Of Hdac2 In Complex With An Inhibitor (Compound 19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZLM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZLM
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Structure Of Hdac2 In Complex With A Macrocyclic Inhibitor (Compound 25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2021-07-14 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, ZL4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-14
Ligands: ZN, SO4, CA, PEG, ZL4
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 20)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, WB4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, PEG, WB4
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Structure Of Human Hdac2 In Complex With Ketone Inhibitor (Compound E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-08-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: ZN, SO4, CA, PEG, V1P
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Structure Of Human Hdac2 In Complex With Ketone Inhibitor (Compound O)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2020-08-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: ZN, SO4, CA, PEG, V1S
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Structure Of Human Hdac2 In Complex With An Aryl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2020-07-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, V1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: ZN, CA, SO4, PEG, V1D
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Co-Structure Of Btk Kinase Domain With L-005085737 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULV, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULV, 5WE
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Co-Structure Of Btk Kinase Domain With L-005191930 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULY, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULY, 5WE
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Co-Structure Of Btk Kinase Domain With L-005298385 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: UM4, EDO, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: UM4, EDO, BTB
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: TV1, ZN, CA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: TV1, ZN, CA, PEG
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor Containing A Spiro-Bicyclic Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: ZN, SO4, CA, PEG, TV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: ZN, SO4, CA, PEG, TV7
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Btk-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-03-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5WH, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-23
Ligands: 5WH, 5WE
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Btk Kinase Domain With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-03 Classification: TRANSFERASE Ligands: 5WF, 5WE, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 5WF, 5WE, CL, EDO
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Discovery Of An Irreversible Hcv Ns5B Polymerase Inhibitor
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2013-12-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2F3, PO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-12-11
Ligands: 2F3, PO4
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Hcv Ns5B Polymerase Complexed With Pyridonylindole Compound
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2013-10-09 Classification: TRANSFERASE Ligands: 8Y6, PO4 |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: 8Y6, PO4
