Search Count: 17
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Cdk2 With Compound 14 Inhibitor With Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-07-07 Classification: SIGNALING PROTEIN, Transferase/Inhibitor Ligands: YOS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: YOS
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Crystal Structure Of Bcl-Xl In Complex With A Benzothiazole-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2021-06-23 Classification: APOPTOSIS Ligands: XZM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-23
Ligands: XZM
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Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYV
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Brd4_Bromodomain2 Complex With Pyrrolopyridone Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYV
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Brd2_Bromodomain2 Complex With Pyrrolopyridone Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYY
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Brd4_Bromodomain1 Complex With Pyrrolopyridone Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2020-05-06 Classification: SIGNALING PROTEIN Ligands: QYY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: QYY
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CJY
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-10-04 Classification: signaling protein/inhibitor Ligands: CN7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: CN7
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Crystal Structure Of Human Nampt With A-1293201
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: 7T7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 7T7, SO4
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Crystal Structure Of Human Nampt With A-1326133
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2017-06-28 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 7TA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: SO4, 7TA
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HY
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Crystal Structure Of Human Nampt With Isoindoline Urea Inhibitor Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8HV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 8HV
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Crystal Structure Of Mcl-1 In Complex With A Bim Competitive Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2017-05-03 Classification: signaling protein/inhibitor Ligands: 9EA, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-03
Ligands: 9EA, ZN
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Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: APOPTOSIS/INHIBITOR Ligands: 3CQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: 3CQ
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Bcl_2-Navitoclax Analog (With Indole) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2014-01-29 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1Y1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-29
Ligands: 1Y1
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Bcl_2-Navitoclax (Abt-263) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-08-14 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1XJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1XJ
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Bcl_2-Navitoclax Analog (Without Thiophenyl) Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-08-14 Classification: APOPTOSIS REGULATOR/INHIBITOR Ligands: 1XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: 1XV
