Search Count: 15
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Mettl3-Mettl14 Heterodimer Bound To The Sam Competitive Small Molecule Inhibitor Stm2457
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2021-04-14 Classification: RNA BINDING PROTEIN Ligands: V22, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-14
Ligands: V22, DMS
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(((3R,4R,5S)-3-((4,4-Difluorocyclohexyl)Methoxy)-5-Methoxypiperidin-4-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XX, SO4
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N-Terminal Bromodomain Of Human Brd4 With 8-(((3R,4R,5S)-3-((4,4-Difluorocyclohexyl)Methoxy)-5-Methoxypiperidin-4-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XX
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N-Terminal Bromodomain Of Human Brd4 With 5-(5-Aminopyridin-3-Yl)-8-(((3R,4R)-3-((1,1-Dioxidotetrahydro-2H-Thiopyran-4-Yl)Methoxy)Piperidin-4-Yl)Amino)-3-Methyl-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XW
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Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-2-(4- Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: N1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: N1D
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Bromodomain Of Human Brd9 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1- Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: TVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: TVU
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Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, XZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, XZB
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Bromodomain Of Human Brd9 With N-(1,1-Dioxo-1-Thian-4-Yl)-5-Ethyl-4- Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C-Pyridine-2- Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, H1B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, H1B
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N-Terminal Bromodomain Of Human Brd4 With 7-(3,4-Dimethoxyphenyl)-N-(1,1-Dioxo-1-Thian-4-Yl)-5-Methyl-4-Oxo-4H,5H-Thieno-3,2-C-Pyridine-2- Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: CA, EDO, TVU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: CA, EDO, TVU
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N-Terminal Bromodomain Of Human Brd4 With N-(1,1-Dioxo-1-Thian-4-Yl)- 5-Methyl-4-Oxo-7-3-(Trifluoromethyl)Phenyl-4H,5H-Thieno-3,2-C- Pyridine-2-Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, 5V2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, 5V2
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N-Terminal Bromodomain Of Human Brd4 With 7-(3,4-Dimethoxyphenyl)-2-(4-Methanesulfonylpiperazine-1-Carbonyl)-5-Methyl-4H,5H-Thieno-3,2-C- Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2015-04-22 Classification: TRANSCRIPTION Ligands: EDO, N1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: EDO, N1D
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With I-Bet151(Gsk1210151A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2011-11-02 Classification: SIGNALING PROTEIN Ligands: EDO, 1GH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: EDO, 1GH
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Crystal Structure Of Novel Protein Emsy Truncate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-10-13 Classification: CHROMATIN REGULATOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-13
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Crystal Structure Of Novel Protein Emsy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2005-10-13 Classification: CHROMATIN REGULATOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-13
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Structure Of The Chromodomain From Mouse Hp1Beta In Complex With The Lysine 9-Methyl Histone H3 N-Terminal Peptide, Nmr, 25 Structures
Organism: Mus musculus
Method: SOLUTION NMR Release Date: 2002-03-12 Classification: CHROMATIN-BINDING |
Organism: Mus musculus
Method: SOLUTION NMR
Release Date: 2002-03-12
