Search Count: 25
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Protac-Mediated Complex Of Kras With Vhl/Elongin-B/Elongin-C/Cullin-2/Rbx1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.50 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: ZN, GDP, WYL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-12-06
Ligands: ZN, GDP, WYL
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Kras-G12C In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: GDP, MG, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, MG, WYU
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Crystal Structure Of Ligand Acbi3 In Complex With Kras G12D C118S Gdp And Pvhl:Elonginc:Elonginb Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2023-12-06 Classification: GENE REGULATION Ligands: PO4, WYL, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: PO4, WYL, GDP, MG
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Crystal Structure Of Compound 3 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: GDP, X4R, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, X4R, MG
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Crystal Structure Of Compound 4 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: X53, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: X53, GDP, MG
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Crystal Structure Of The Vcb Complex With Compound 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2023-05-31 Classification: LIGASE Ligands: WBN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: WBN, CL
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Beta-Catenin In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2020-12-16 Classification: ONCOPROTEIN Ligands: R9Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: R9Q
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Crystal Structure Of Crystal Form 2 Of An Active Kras G12D (Gppcp) Dimer In Complex With Bi-5747
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2020-11-18 Classification: SIGNALING PROTEIN Ligands: MG, GCP, R6W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: MG, GCP, R6W
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Egfr-Kinase In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2019-11-20 Classification: TRANSFERASE Ligands: L1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: L1H
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Egfr-Kinase In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2019-11-20 Classification: TRANSFERASE Ligands: L1K, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: L1K, DMS
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Egfr-Kinase In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2019-11-20 Classification: TRANSFERASE Ligands: L3Z, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: L3Z, DMS
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Crystal Structure Phgdh In Complex With Nadh And 3-Phosphoglycerate At 1.77 A Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: 3PG, NAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: 3PG, NAI
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Crystal Structure Of Phgdh In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: K4T, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: K4T, SO4
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Crystal Structure Of Phgdh In Complex With Compound 40
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: SO4, K52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K52
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Crystal Structure Of Phgdh In Complex With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: SO4, K58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K58
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Crystal Structure Of Phgdh In Complex With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: SO4, K5N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: SO4, K5N
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Crystal Structure Of Phgdh In Complex With Bi-4924
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-08-07 Classification: OXIDOREDUCTASE Ligands: K5K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-07
Ligands: K5K
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: GCP, MG, F0N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GCP, MG, F0N
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: MG, NO3, GCP, EZZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: MG, NO3, GCP, EZZ
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Crystal Structure Of Kras G12D (Gppcp) In Complex With 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2019-07-31 Classification: SIGNALING PROTEIN Ligands: MG, GCP, F0B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: MG, GCP, F0B
