Search Count: 20
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Discovery Of A Highly Potent And Broadly Effective Egfr And Her2 Exon 20 Insertion Mutant Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2018-07-18 Classification: Transferase/Transferase Inhibitor Ligands: FZP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-18
Ligands: FZP
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Crystal Structure Of Dipeptidyl Peptidase Iv In Complex With Syr-472
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-07-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 6RL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-13
Ligands: NAG, 6RL
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Renin In Complexed With 4-Methoxy-3-(3-Methoxypropoxy)-N-{[(3S,4S)-4-{[(4-Methylphenyl)Sulfonyl]Amino}Pyrrolidin-3-Yl]Methyl}-N-(Propan-2-Yl)Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2015-03-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 3ZK, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: NAG, 3ZK, SO4, DMS
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Renin In Complexed With N-({(3S,4S)-4-[(Benzylsulfonyl)Amino]Pyrrolidin-3-Yl}Methyl)-4-Methoxy-3-(3-Methoxypropoxy)-N-(Propan-2-Yl)Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-03-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 3ZJ, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: NAG, 3ZJ, SO4, DMS
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Renin In Complexed With (3S,4S)-4-({[4-Methoxy-3-(3-Methoxypropoxy)Benzoyl](Propan-2-Yl)Amino}Methyl)Pyrrolidin-3-Yl Benzylcarbamate Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-03-25 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 3ZN, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: NAG, 3ZN, SO4, DMS
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Crystal Structure Of Rock 1 Bound To Yb-15-Qd37
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3J7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 3J7
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Crystal Structure Of Renin In Complex With Compound4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2014-10-08 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 2XF, DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: NAG, 2XF, DMS, SO4
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Structure-Based Design Of 4-Hydroxy-3,5-Substituted Piperidines As Direct Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2014-08-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DMS, NAG, PO4, 2Y9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: DMS, NAG, PO4, 2Y9
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Crystal Structure Of Renin In Complex With Nvp-Amq838 (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-03-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAG, 0LR
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Crystal Structure Of Renin In Complex With Nvp-Ayz832 (Compound 6A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2013-03-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAG, 0LS, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bca079 (Compound 12A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-03-06 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAG, 0LT, SO4
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Crystal Structure Of Renin In Complex With Pkf909-724 (Compound 3)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0LU, SO4, 0LW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0LU, SO4, 0LW
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Crystal Structure Of Renin In Complex With Gp055321 (Compound 4)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0M2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0M2
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Crystal Structure Of Renin In Complex With Nvp-Ayl747 (Compound 5)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0M3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0M3, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bbv031 (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0ME, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0ME, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bch965 (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0MJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0MJ, SO4
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Crystal Structure Of Renin In Complex With Nvp-Bgq311 (Compound 12)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2013-02-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 0N0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-13
Ligands: NAG, 0N0, SO4
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Crystal Structure Of Human Dpp4 Bound To Tak-294
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2011-10-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: LUI, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: LUI, NAG
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Crystal Structure Of Human Dpp4 Bound To Tak-986
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2011-02-09 Classification: HYDROLASE,SIGNALING PROTEIN/INHIBITOR Ligands: 10T, NAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-09
Ligands: 10T, NAG
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Crystal Structure Of Human Dpp4 Bound To Tak-100
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2011-01-26 Classification: HYDROLASE,SIGNALING PROTEIN/INHIBITOR Ligands: NAG, 01T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-01-26
Ligands: NAG, 01T