Search Count: 20
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2022-03-23 Classification: TRANSFERASE/INHIBITOR Ligands: SAM, 7U2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-23
Ligands: SAM, 7U2
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2022-03-23 Classification: TRANSFERASE/INHIBITOR Ligands: SAM, CL, EDO, PEG, 7UB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-23
Ligands: SAM, CL, EDO, PEG, 7UB
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"Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Agi-43192
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.97 Å Release Date: 2022-03-23 Classification: TRANSFERASE/INHIBITOR Ligands: SAM, CL, EDO, 7UN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-23
Ligands: SAM, CL, EDO, 7UN, GOL
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Agi-41998
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2022-03-23 Classification: TRANSFERASE/INHIBITOR Ligands: SAM, 7UI, EDO, GOL, 1PE, CL, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-23
Ligands: SAM, 7UI, EDO, GOL, 1PE, CL, MG
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Ag-270
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: CL, EDO, SAM, WBG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: CL, EDO, SAM, WBG
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: J41, SAM, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: J41, SAM, CL
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Agi-24512
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: J4A, SAM, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: J4A, SAM, EDO, GOL
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: SAM, CL, TRS, GOL, WBM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: SAM, CL, TRS, GOL, WBM
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Crystal Structure Of Human Methionine Adenosyltransferase 2A (Mat2A) In Complex With Sam And Allosteric Inhibitor Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: WBS, CL, TRS, EDO, GOL, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: WBS, CL, TRS, EDO, GOL, SAM
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Crystal Structure Of Human Cytosolic Isocitrate Dehydrogenase (Idh1) R132H Mutant In Complex With Nadph And Ag-881 (Vorasidenib) Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2020-02-05 Classification: ANTITUMOR PROTEIN Ligands: NDP, SO4, 33O, PEG, ACT, MLA, 9UO, MLT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: NDP, SO4, 33O, PEG, ACT, MLA, 9UO, MLT
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Crystal Structure Of Human Mitochondrial Isocitrate Dehydrogenase (Idh2) R140Q Mutant Homodimer In Complex With Nadph And Ag-881 (Vorasidenib) Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2020-02-05 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: 9UO, NDP, CA, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: 9UO, NDP, CA, NA
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Crystal Structure Of Human Cytosolic Isocitrate Dehydrogenase (Idh1) R132H Mutant In Complex With Nadph And Agi-15056
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2020-02-05 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: NDP, QWM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-05
Ligands: NDP, QWM
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Crystal Structure Of Human Mitochondrial Isocitrate Dehydrogenase (Idh2) R140Q Mutant Homodimer In Complex With Ag-221 (Enasidenib) Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2017-03-08 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: CA, GOL, NDP, NA, ACT, 69Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-08
Ligands: CA, GOL, NDP, NA, ACT, 69Q
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Crystal Structure Of Human Mitochondrial Isocitrate Dehydrogenase R140Q Mutant Homodimer Bound To Nadph And Alpha-Ketoglutaric Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2017-03-01 Classification: OXIDOREDUCTASE Ligands: NDP, CA, GOL, ACT, AKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: NDP, CA, GOL, ACT, AKG
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2011-11-02 Classification: TRANSFERASE/transferase inhibitor Ligands: BOG, P5K |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-11-02
Ligands: BOG, P5K
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P78 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P78
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P79 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P79
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P7A |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P7A
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: P7B, BOG |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: P7B, BOG
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P38 Inhibitor-Bound
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-10-12 Classification: transferase/transferase inhibitor Ligands: BOG, P7C |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2011-10-12
Ligands: BOG, P7C
