Search Count: 23
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Mtb Guab Dcbs In Complex With Inhibitor G1
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-27 Classification: OXIDOREDUCTASE Ligands: IMP, VOA, SO4 |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: IMP, VOA, SO4
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Mtb Guab Dcbs In Complex With Inhibitor Compound 5
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-11-27 Classification: OXIDOREDUCTASE Ligands: IMP, A1A3K |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: IMP, A1A3K
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E. Coli Msba In Complex With Lps And Inhibitor G7090 (Compound 3)
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2022-03-09 Classification: TRANSLOCASE Ligands: 95X, KDL |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2022-03-09
Ligands: 95X, KDL
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E. Coli Lepb In Complex With Gne0775 ((4S,7S,10S)-10-((S)-4-Amino-2-(2-(4-(Tert-Butyl)Phenyl)-4-Methylpyrimidine-5-Carboxamido)-N-Methylbutanamido)-16,26-Bis(2-Aminoethoxy)-N-(2-Iminoethyl)-7-Methyl-6,9-Dioxo-5,8-Diaza-1,2(1,3)-Dibenzenacyclodecaphane-4-Carboxamide)
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2018-10-10 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: CZD, 1PE |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: CZD, 1PE
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E. Coli Msba In Complex With Lps And Inhibitor G907
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2018-05-02 Classification: LIPID TRANSPORT Ligands: 3PE, AU7, FTT, PA1, PO4, DAO, MYR, DPO |
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: 3PE, AU7, FTT, PA1, PO4, DAO, MYR, DPO
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E. Coli Msba In Complex With Lps And Inhibitor G092
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2018-05-02 Classification: LIPID TRANSPORT Ligands: E1M, FTT, DAO, 3PE, PO4, MYR |
Organism: Escherichia coli o6:h1 (strain cft073 / atcc 700928 / upec)
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: E1M, FTT, DAO, 3PE, PO4, MYR
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Cdk8/Cycc In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-04-20 Classification: Transferase/Transcription Ligands: 66X, FMT, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: 66X, FMT, CL
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Crystal Structure Of Cdk8:Cyclin C Complex With Compound 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-02-10 Classification: Transcription/Transferase/Inhibitor Ligands: EDO, FMT, 50R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: EDO, FMT, 50R
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Discovery Of A Potent And Selective Bcl-Xl Inhibitor That Demonstrates Thrombocytopenia And Inhibits Tumor Growth In Vivo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-07-22 Classification: APOPTOSIS/INHIBITOR Ligands: 3CQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-22
Ligands: 3CQ
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Bcl-Xl In Complex With Inhibitor (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-10-15 Classification: APOPTOSIS Ligands: 38H, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-15
Ligands: 38H, EDO, ACT
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Jak2 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-[(8As)-2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(8Ah)-Yl]Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexanecarbonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J5
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Jak1 Kinase (Jh1 Domain) In Complex With The Inhibitor (Trans-4-{2-[(1R)-1-Hydroxyethyl]Imidazo[4,5-D]Pyrrolo[2,3-B]Pyridin-1(6H)-Yl}Cyclohexyl)Acetonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1J6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 1J6
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 34
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2013-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 15T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 15T
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The Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2012-07-04 Classification: Transferase/Transferase Inhibitor Ligands: JAK, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK, EDO
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Jak1 Kinase (Jh1 Domain) In Complex With Compound 20
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 0Q2
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Discovery And Optimization Of C-2 Methyl Imidazo-Pyrrolopyridines As Potent And Orally Bioavailable Jak1 Inhibitors With Selectivity Over Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.82 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1RS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: 1RS
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Discovery And Optimization Of C-2 Methyl Imidazo-Pyrrolopyridines As Potent And Orally Bioavailable Jak1 Inhibitors With Selectivity Over Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: JAK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: JAK
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Crystal Structure Of Bcl-Xl In Complex With A Quinazoline Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2011-04-06 Classification: APOPTOSIS/INHIBITOR Ligands: HI0, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-04-06
Ligands: HI0, CL, GOL
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Structure Of An Ml-Iap/Xiap Chimera Bound To A Peptidomimetic
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2010-03-09 Classification: APOPTOSIS Ligands: ZN, 516 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: ZN, 516