Search Count: 13
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Discovery Of Oral Polo-Like Kinase (Plk) Inhibitors With Enhanced Selectivity Profile Using Residue Targeted Drug Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-08-21 Classification: TRANSFERASE Ligands: 9ZP, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-21
Ligands: 9ZP, SO4
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Choline Kinase Alpha Acts Through A Double-Displacement Kinetic Mechanism Involving Enzyme Isomerisation, As Determined Through Enzyme And Inhibitor Kinetics And Structural Biology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-04-17 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 0H7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: SO4, 0H7
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Crystal Structure Of Itk Kinase Bound To An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-06-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PQC, L7A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: PQC, L7A
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Crystal Structure Of Itk Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-06-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PQC, L7O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-22
Ligands: PQC, L7O
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Crystal Structure Of Aurora-2, An Oncogenic Serine-Threonine Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2003-04-15 Classification: TRANSFERASE Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-04-15
Ligands: ADN
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Complex Of A Y195F Mutant Cgtase From B. Circulans Strain 251 Complexed With A Maltononaose Inhibitor At Ph 9.8 Obtained After Soaking The Crystal With Acarbose And Maltohexaose
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 1998-12-09 Classification: GLYCOSYLTRANSFERASE Ligands: CA, ADH |
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION
Release Date: 1998-12-09
Ligands: CA, ADH
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Cyclodextrin Glycosyltransferase W616A Mutant From Bacillus Circulans Strain 251
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1997-04-21 Classification: GLYCOSYLTRANSFERASE Ligands: CA |
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION
Release Date: 1997-04-21
Ligands: CA
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Thermostable Cgtase From Thermoanaerobacterium Thermosulfurigenes Em1 At Ph 8.0.
Organism: Thermoanaerobacterium thermosulfurigenes
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 1996-03-08 Classification: GLYCOSIDASE Ligands: CA |
Organism: Thermoanaerobacterium thermosulfurigenes
Method: X-RAY DIFFRACTION
Release Date: 1996-03-08
Ligands: CA
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Complex Of Cgtase With Maltotetraose At Room Temperature And Ph 9.1 Based On Diffraction Data Of A Crystal Soaked With Alpha-Cyclodextrin
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 1995-12-15 Classification: GLYCOSYLTRANSFERASE Ligands: CA |
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION
Release Date: 1995-12-15
Ligands: CA
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Complex Of A (D229N/E257Q) Double Mutant Cgtase From Bacillus Circulans Strain 251 With Maltotetraose At 120 K And Ph 9.1 Obtained After Soaking The Crystal With Alpha-Cyclodextrin
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 1995-12-15 Classification: GLYCOSYLTRANSFERASE Ligands: CA |
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION
Release Date: 1995-12-15
Ligands: CA
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Complex Of Cgtase With Maltotetraose At Room Temperature And Ph 9.6 Based On Diffraction Data Of A Crystal Soaked With Maltoheptaose
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 1995-12-15 Classification: GLYCOSYLTRANSFERASE Ligands: CA |
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION
Release Date: 1995-12-15
Ligands: CA
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Wild-Type Cgtase From Bacillus Circulans Strain 251 At 120 K And Ph 7.55
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 1995-12-15 Classification: GLYCOSYLTRANSFERASE Ligands: CA |
Organism: Bacillus circulans
Method: X-RAY DIFFRACTION
Release Date: 1995-12-15
Ligands: CA
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The Solution Structure Of The Human Retinoic Acid Receptor-Beta Dna-Binding Domain
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 1994-01-31 Classification: DNA-BINDING RECEPTOR Ligands: ZN |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 1994-01-31
Ligands: ZN
