Search Count: 11
![]() |
Mers Mpro With Egt710
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION Resolution:3.04 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1CBU |
Organism: Middle east respiratory syndrome-related coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1CBU
![]() |
Oc43 Mpro With Egt710
Organism: Human coronavirus oc43
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1CBU |
Organism: Human coronavirus oc43
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1CBU
![]() |
Lipid A Secondary Acyltransferase Lpxm From Acinetobacter Baumannii
Organism: Acinetobacter baumannii niph 410
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-09-28 Classification: TRANSFERASE Ligands: SO4, NA, GOL, LMT, PO4 |
Organism: Acinetobacter baumannii niph 410
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: SO4, NA, GOL, LMT, PO4
![]() |
Lipid A Secondary Acyltransferase Lpxm From Acinetobacter Baumannii With Catalytic Residue Substitution (E127A)
Organism: Acinetobacter baumannii niph 410
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-09-28 Classification: TRANSFERASE Ligands: SO4, GOL, LMT, 11A |
Organism: Acinetobacter baumannii niph 410
Method: X-RAY DIFFRACTION
Release Date: 2016-09-28
Ligands: SO4, GOL, LMT, 11A
![]() |
Co-Crystal Structure Of Lipid Kinase Pi3K Alpha With A Selective Phosphatidylinositol-3 Kinase Alpha Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-05-18 Classification: transferase/transferase inhibitor Ligands: 4Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 4Q2
![]() |
Discovery Of Imidazo[1,2-A]-Pyridine Inhibitors Of Pan-Pi3 Kinases That Are Efficacious In A Mouse Xenograft Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 5XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: GOL, 5XV
![]() |
The Crystal Structure Of Human Vps34 In Complex With Pik-Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-10-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 2UG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-29
Ligands: GOL, 2UG
![]() |
Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UJ, SO4
![]() |
Structure Of Pi3K Gamma With Imidazopyridine Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2013-07-17 Classification: Transferase/Transferase Inhibitor Ligands: 1UK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-17
Ligands: 1UK, SO4
![]() |
Crystal Structure Of Pi3K Gamma With N6-(3,4-Dimethoxyphenyl)-2-Morpholino-[4,5'-Bipyrimidine]-2',6-Diamine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-08-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 13K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 13K, SO4
![]() |
Crystal Structure Of Pi3K Gamma With 3-(2-Morpholino-6-(Pyridin-3-Ylamino)Pyrimidin-4-Yl)Phenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2011-08-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P2B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: P2B
