Search Count: 18
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Discovery Of Potent And Efficacious Cyanoguanidine-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: LTS, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: LTS, PO4, EDO
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Discovery Of Potent And Efficacious Cyanoguanidine-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2013-12-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: LWW, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-12-25
Ligands: LWW, PO4, EDO
 |
Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20J, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20J, PO4, EDO
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Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20M, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20M, PO4, EDO
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Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20N, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20N, PO4, EDO
 |
Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, 1EB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: PO4, 1EB, EDO
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Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20P, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20P, PO4, EDO
 |
Fragment-Based Identification Of Amides Derived From Trans-2-(Pyridin-3-Yl)Cyclopropanecarboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20O, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20O, PO4, EDO
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Identification Of Amides Derived From 1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20R, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20R, PO4
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Identification Of Amides Derived From 1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid As Potent Inhibitors Of Human Nicotinamide Phosphoribosyltransferase (Nampt)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2013-09-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 20T, POP, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: 20T, POP, PO4
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Discovery Of Potent And Efficacious Urea-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors With Reduced Cyp2C9 Inhibition Properties
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-05-29 Classification: Transferase/Transferase inhibitor Ligands: 1LJ, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-29
Ligands: 1LJ, PO4, EDO
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Structure-Based Identification Of Ureas As Novel Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2013-05-08 Classification: Transferase/Transferase inhibitor Ligands: 1LS, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-08
Ligands: 1LS, PO4, EDO
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Structure-Based Discovery Of Novel Amide-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2013-05-08 Classification: Transferase/Transferase Inhibitor Ligands: 1QR, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-08
Ligands: 1QR, PO4, EDO
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Structure-Based Discovery Of Novel Amide-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2013-05-08 Classification: Transferase/transferase Inhibitor Ligands: 1QS, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-08
Ligands: 1QS, PO4, EDO
 |
Phd2-R127 With Jnj41536014
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2010-12-01 Classification: OXIDOREDUCTASE Ligands: FE2, SO4, 014 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: FE2, SO4, 014
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Phd2-R717 With 40787422
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2010-12-01 Classification: OXIDOREDUCTASE Ligands: ACT, FE2, 42Z, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: ACT, FE2, 42Z, PEG
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Phd2 With 2-Oxoglutarate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-12-01 Classification: OXIDOREDUCTASE Ligands: SO4, FE2, AKG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-01
Ligands: SO4, FE2, AKG
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The Structure Of A Class Ii Ubiquitin-Conjugating Enzyme, Ubc1.
Organism: Saccharomyces cerevisiae
Method: SOLUTION NMR Release Date: 2004-08-31 Classification: LIGASE |
Organism: Saccharomyces cerevisiae
Method: SOLUTION NMR
Release Date: 2004-08-31