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8ETR image
Cryoem Structure Of Nlrp3 Nacht Domain In Complex With G2394

7MSA image
Gdc-9545 In Complex With Estrogen Receptor Alpha

7KHH image
Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)

7KHL image
Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.29 Å Release Date: 2021-02-24
Classification: CELL CYCLE
Ligands: WEM, GOL

6WOK image
Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 6

6PET image
Crystal Structure Of 8-Hydroxychromene Compound 30 Bound To Estrogen Receptor Alpha

6PFM image
Crystal Structure Of Gdc-0927 Bound To Estrogen Receptor Alpha

6DF6 image
Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 16Ab

6DFN image
Crystal Structure Of Estrogen Receptor Alpha In Complex With Receptor Degrader 16Aa

5WHC image
Usp7 In Complex With Cpd2 (4-(3-(1-Methylpiperidin-4-Yl)-1,2,4-Oxadiazol-5-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2017-12-13
Classification: HYDROLASE
Ligands: AJJ, GOL

5UQV image
Usp7 In Complex With Gne6640 (4-(2-Amino-4-Ethyl-5-(1H-Indazol-5-Yl)Pyridin-3-Yl)Phenol)

5UQX image
Usp7 In Complex With Gne6776 (6'-Amino-4'-Ethyl-5'-(4-Hydroxyphenyl)-N-Methyl-[3,3'-Bipyridine]-6-Carboxamide)

5KTU image
Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.38 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XB, DMS

5KTW image
Crebbp Bromodomain In Complex With Cpd 44 (3-((5-Acetyl-1-(Cyclopropylmethyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[4,3-C]Pyridin-3-Yl)Amino)-N-Isopropylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.09 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XG, EDO

5KTX image
Crebbp Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.27 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: 6XH, EDO, DMS

5KU3 image
Brd4 Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.14 Å Release Date: 2016-11-02
Classification: TRANSFERASE
Ligands: EDO, DMS, GOL, PEG, 6XH

3H0Y image
Aurora A In Complex With A Bisanilinopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2009-07-07
Classification: TRANSFERASE
Ligands: 48B, SO4

3H0Z image
Aurora A In Complex With A Bisanilinopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.92 Å Release Date: 2009-07-07
Classification: TRANSFERASE
Ligands: 45B
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