Search Count: 26
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C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, SO4
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 98A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 98A
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9XO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9XO
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9OO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9OO
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9VV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9VV
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: EDO, 9WU, BR, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: EDO, 9WU, BR, CL
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9KI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9KI
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C-Kit T670I Mutated Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI
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Pdgfra T674I Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, PEG
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Pdgfra T674I Mutant Kinase Domain In Complex With Avapritinib Derivative 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9OO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9OO, PEG
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Pdgfra Wild-Type Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2023-12-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
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Apo Crystal Structure Of Pdgfra-T674I Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-12-27 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
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Crystal Structure Of Egfr-T790M/C797S In Complex With Brigatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2023-05-03 Classification: TRANSFERASE Ligands: 6GY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: 6GY
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Crystal Structure Of Egfr-T790M/C797S In Complex With Wz4002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-05-03 Classification: TRANSFERASE Ligands: 0UN, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: 0UN, MES
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Crystal Structure Of Egfr-T790M/C797S In Complex With Reversible Aminopyrimidine 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2023-05-03 Classification: TRANSFERASE Ligands: R25, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: R25, MES
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Crystal Structure Of Egfr-T790M/V948R In Complex With Reversible Aminopyrimidine 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-05-03 Classification: TRANSFERASE Ligands: V58, SO4, CL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: V58, SO4, CL, NA
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Protein Kinase Mkk7 In Complex With Phenethyltriazole-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 2GI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 2GI
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Protein Kinase Mkk7 In Complex With Difluoro-Phenethyltriazole-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 24N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 24N
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Protein Kinase Mkk7 In Complex With 5-Bromo-2-Hydroxyphenyl-Substituted Pyrazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: GOL, 2I5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: GOL, 2I5
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Protein Kinase Mkk7 In Complex With Methoxycyclohexyl-Substituted Indazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2022-07-20 Classification: TRANSFERASE Ligands: 1XZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-20
Ligands: 1XZ
