Search Count: 43
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Crystal Structure Of Plekha7 Ph Domain Biding So4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2021-04-07 Classification: CELL ADHESION Ligands: SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: SO4, GOL
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Crystal Structure Of Plekha7 Ph Domain Biding Inositol-Tetraphosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2021-04-07 Classification: CELL ADHESION Ligands: 4IP, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: 4IP, EDO
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Crystal Structure Of Ligand-Free Plekha7 Ph Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2021-04-07 Classification: CELL ADHESION Ligands: GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: GOL, EDO
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Cocomplex Structure Of Deoxyhypusine Synthase With Inhibitor 6-[(1R)-2-Amino-1-Phenylethyl]-3-(Pyridin-3-Yl)-4H,5H,6H,7H-Thieno[2,3-C]Pyridin-7-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2020-08-19 Classification: TRANSFERASE/INHIBITOR Ligands: 8Y1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: 8Y1
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Cocomplex Structure Of Deoxyhypusine Synthase With Inhibitor 6-[(2R)-1-Amino-4-Methylpentan-2-Yl]-3-(Pyridin-3-Yl)-4H,5H,6H,7H-Thieno[2,3-C]Pyridin-7-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2020-08-19 Classification: TRANSFERASE/INHIBITOR Ligands: 91A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: 91A
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1.65 Angstrom Ternary Complex Of Deoxyhypusine Synthase With Cofactor Nad And Spermidine Mimic Inhibitor Gc7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: NAD, GC7, MPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: NAD, GC7, MPD
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Cocomplex Structure Of Deoxyhypusine Synthase With Inhibitor 6-Bromo-N-(1H-Indol-4-Yl)-1-Benzothiophene-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: 8XY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: 8XY
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KAV
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KA4
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KA7
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Structure Of Cdk12/Cyck In Complex With A Small Molecule Inhibitor N-(4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)-N-((1R,4R)-4-(Quinazolin-2-Ylamino)Cyclohexyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-08-29 Classification: TRANSFERASE/INHIBITOR Ligands: MG, 8M1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: MG, 8M1
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Structure Of Cdc2-Like Kinase 2 (Clk2) In Complex With Compound T-025 [N2-Methyl-N4-(Pyrimidin-2-Ylmethyl)-5-(Quinolin-6-Yl)-7H-Pyrrolo[2,3-D]Pyrimidine-2,4-Diamine]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.92 Å Release Date: 2018-05-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8FY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-09
Ligands: 8FY
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Crystal Structure Of Human Brr2 In Complex With T-3905516
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-07-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, 8LS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: GOL, 8LS
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Crystal Structure Of Human Brr2 In Complex With T-3935799
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2017-07-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, 8LP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: GOL, 8LP
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Crystal Structure Of Human Brr2 In Complex With T-1206548
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-07-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 8LV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: 8LV
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Crystal Structure Of Autotaxin/Enpp2 With A Covalent Fragment
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-03-15 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, NAG, ACT, 6C1 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: ZN, CA, NAG, ACT, 6C1
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Human Givd Cytosolic Phospholipase A2 In Complex With Methyl Gamma-Linolenyl Fluorophosphonate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2016-06-08 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 7FA, BA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 7FA, BA
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Human Givd Cytosolic Phospholipase A2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-06-08 Classification: HYDROLASE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: SO4
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Human Givd Cytosolic Phospholipase A2 In Complex With Methyl Gamma-Linolenyl Fluorophosphonate Inhibitor And Terbium Chloride
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2016-06-08 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 7FA, TB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 7FA, TB
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Structure Of Protein Kinase C Theta With Compound 10: 2,2-Dimethyl-7-(2-Oxidanylidene-3~{H}-Imidazo[4,5-B]Pyridin-1-Yl)-1-(Phenylmethyl)-3~{H}-Quinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-05-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5VS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-11
Ligands: 5VS
