Search Count: 18
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Kdm2A-Nucleosome Structure Stabilized By H3K36C-Unc8015 Covalent Conjugate
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2023-02-22 Classification: GENE REGULATION/DNA Ligands: OH0, FE |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2023-02-22
Ligands: OH0, FE
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Crystal Structure Of Kdm2A Histone Demethylase Catalytic Domain In Complex With An H3C36 Peptide Modified By Unc8015
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2023-02-22 Classification: GENE REGULATION Ligands: FE, OH0 |
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: FE, OH0
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Structure Of Vrk1 C-Terminal Tail Bound To Nucleosome Core Particle
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Release Date: 2022-05-04 Classification: STRUCTURAL PROTEIN/DNA/TRANSFERASE |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2022-05-04
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Mrt10241866A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-05-05 Classification: TRANSFERASE Ligands: Y6V, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: Y6V, UNX
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Unc6934
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: V01, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: V01, UNX
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc3437
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2019-09-11 Classification: Transferase/Transferase Inhibitor Ligands: CL, 9VS, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-11
Ligands: CL, 9VS, MG
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc2541
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-02-22 Classification: Transferase/Transferase Inhibitor Ligands: CL, K0X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: CL, K0X
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc2434
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2017-01-11 Classification: Transferase/Transferase Inhibitor Ligands: CL, 6Q1, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: CL, 6Q1, MG
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc1896
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2014-05-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, MG, MH7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
Ligands: CL, MG, MH7
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc1817
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2014-05-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, 4MH, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-05-21
Ligands: CL, 4MH, MG
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc1917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2013-11-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, MG, 24K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-27
Ligands: CL, MG, 24K
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Crystal Structure Of The 3-Mbt Repeat Domain Of L3Mbtl3 And Unc2533 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2013-07-10 Classification: TRANSCRIPTION Ligands: 1VZ, SO4, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 1VZ, SO4, UNX
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Crystal Structure Of The Complex Of The 3-Mbt Repeat Domain Of L3Mbtl3 And Unc1215
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2012-06-27 Classification: TRANSCRIPTION Ligands: UWN, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-27
Ligands: UWN, UNX
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Crystal Structure Of The Catalytic Domain Of The Proto-Oncogene Tyrosine-Protein Kinase Mer In Complex With Inhibitor Unc569
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2012-06-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CKJ, CL, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-20
Ligands: CKJ, CL, CA
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The 3-Mbt Repeat Domain Of L3Mbtl1 In Complex With A Methyl-Lysine Mimic
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-03-07 Classification: TRANSCRIPTION Ligands: UWN, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-07
Ligands: UWN, UNX
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Crystal Structure Of Histone Lysine Methyltransferase G9A With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2011-05-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAH, CIQ, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-04
Ligands: ZN, SAH, CIQ, UNX
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Crystal Structure Of L3Mbtl1 (Mbt Repeat) In Complex With A Nicotinamide Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2010-11-03 Classification: TRANSCRIPTION Ligands: P8H, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-11-03
Ligands: P8H, SO4, GOL
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Discovery Of A 2,4-Diamino-7-Aminoalkoxy-Quinazoline As A Potent Inhibitor Of Histone Lysine Methyltransferase, G9A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: ZN, SAH, DXQ, CL, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: ZN, SAH, DXQ, CL, UNX
