Search Count: 29
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365096A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-03-13 Classification: HYDROLASE Ligands: WTE |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-03-13
Ligands: WTE
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365097A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: WTV, GOL, CL |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WTV, GOL, CL
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365096A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: A1ADS |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: A1ADS
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Sara Cov-2 3C-Like Protease In Complex With Gsk3487016A
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: WYR, EDO |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WYR, EDO
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3735967A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, I67, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, I67, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3543105A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, ZN, EDO, GOL, IO5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: SAH, ZN, EDO, GOL, IO5
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830334A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, ZN, GOL, 96I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: EDO, ZN, GOL, 96I
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3852279B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, EDO, GOL, C79 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, EDO, GOL, C79
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Cofactor Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2022-03-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-03-30
Ligands: ZN, SAM, GOL, EDO
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-07-07 Classification: TRANSFERASE Ligands: SAH, ZN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: SAH, ZN, EDO, GOL
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3830052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, X52 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, X52
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Human Dnmt1(729-1600) Bound To Zebularine-Containing 12Mer Dsdna And Inhibitor Gsk3685032A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-07-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR/DNA Ligands: ZN, EDO, UXM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-07
Ligands: ZN, EDO, UXM
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Rip2 Kinase Catalytic Domain Complex With 2(4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl)Oxy)Ethyl Phosphate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: K9T, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: K9T, CA
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Rip2 Kinase Catalytic Domain Complex With 2({4[(1,3Benzothiazol5Yl)Amino]6(2Methylpropane2Sulfonyl)Quinazolin7Yl}Oxy)Ethan1Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2019-07-17 Classification: TRANSFERASE Ligands: KA2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: KA2
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Crystal Structure Of Rip1 Kinase In Complex With A Pyrrolidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2019-05-08 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: M5J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: M5J, SO4
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Crystal Structure Of Rip1 Kinase In Complex With Dhp77
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: JSW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: JSW
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Rip1 Kinase ( Flag 1-294, C34A, C127A, C233A, C240A) With Gsk772
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-07-05 Classification: transferase/transferase inhibitor Ligands: 7MJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: 7MJ
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Compound 3 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GE, SO4
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The Identification And Pharmacological Characterization Of 6-(Tert-Butylsulfonyl)-N-(5-Fluoro-1H-Indazol-3-Yl)Quinolin-4-Amine (Gsk583), A Highly Potent And Selective Inhibitor Of Rip2 Kinase, Gsk583 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 6GD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 6GD
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Crystal Structure Of Rip1 Kinase With A Benzo[B][1,4]Oxazepin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2016-03-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 65U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: 65U