Search Count: 24
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Crystal Structure Of Polo Box Domain In Complex With Cyclic Peptide Inhibitor
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2022-03-02 Classification: TRANSFERASE/Inhibitor |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2022-03-02
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZF
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZL
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZO, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZO, MG
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: FZR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: FZR
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: G0U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: G0U
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Crystal Structure Of Ttk Kinase Domain In Complex With Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2021-05-12 Classification: TRANSFERASE Ligands: G5C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: G5C
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg056
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2019-03-06 Classification: TRANSCRIPTION/INHIBITOR Ligands: X27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-06
Ligands: X27
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Src Kinase Bound To Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-02-27 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6H3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3
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Crystal Structure Of Erk2 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: SO4, 6H3, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: SO4, 6H3, EDO, CL
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Crystal Structure Of Erk1 Covalently Bound To Sm1-71
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2019-02-27 Classification: TRANSFERASE Ligands: 6H3, EWH, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-27
Ligands: 6H3, EWH, SO4, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Xmd17-26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2019-01-16 Classification: TRANSCRIPTION/INHIBITOR Ligands: R4L, EDO, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: R4L, EDO, NO3
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Crystal Structure Of Ack1 With Compound 10D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2018-09-26 Classification: TRANSFERASE Ligands: 9KO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-26
Ligands: 9KO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg046
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.23 Å Release Date: 2018-08-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: EX1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: EX1, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg047
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2018-08-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: X26, EDO, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: X26, EDO, NO3
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg069
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2018-08-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: F3J, EDO, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: F3J, EDO, NO3
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Jwg071
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2018-08-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: F2S, FND, EDO, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: F2S, FND, EDO, NO3
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Inhibitor Xmd11-50
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2018-07-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 4K4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-07-04
Ligands: 4K4, EDO
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Crystal Structure Of Aurora-A In Complex With Fmf-03-145-1 (Compound 2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: 9YQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: 9YQ
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Crystal Structure Of Human Trap1 With Amppnp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2015-04-29 Classification: CHAPERONE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: ANP, MG
