Search Count: 70
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Crystal Structure Of The Hpk1 Kinase Domain In Complex With Inhibitor 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1KCT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1KCT, EDO
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Crystal Structure Of The Hpk1 Kinase Domain In Complex With Inhibitor 6B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1KCQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1KCQ, EDO
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Crystal Structure Of The Hpk1 Kinase Domain In Complex With Inhibitor 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1KCR, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1KCR, EDO
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Sos1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2026-06-24 Classification: SIGNALING PROTEIN Ligands: A1JWK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-24
Ligands: A1JWK
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Structure Of Sos1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2025-09-17 Classification: CYTOSOLIC PROTEIN Ligands: A1I6H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: A1I6H
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITC
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITA
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Pyrazine Carboxamide Inhibitor Az3246 (Compound 24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITB, EDO
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ7
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ8, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: A1IZ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IZ9
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: Q6K, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: Q6K, SO4
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Highly Optimized Cns Penetrant Inhibitors Of Egfr Exon20 Insertion Mutations. Compound 51 Bound To Egfrinsnpg [V948R]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-02-05 Classification: SIGNALING PROTEIN Ligands: A1IUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-05
Ligands: A1IUK
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-07-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, PQI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: MG, GDP, PQI
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2023-07-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, PUO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-12
Ligands: MG, GDP, PUO
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2022-04-20 Classification: SIGNALING PROTEIN Ligands: V4T, MG, GDP, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: V4T, MG, GDP, CA
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2022-04-20 Classification: SIGNALING PROTEIN Ligands: MG, GDP, V52, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: MG, GDP, V52, CA
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Krasg12C Ligand Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2022-04-20 Classification: SIGNALING PROTEIN Ligands: MG, GDP, VLE, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-04-20
Ligands: MG, GDP, VLE, CA
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Crystal Structure Of The Kinase Domain Of Human C-Kit In Complex With A Type-Ii Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.38 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O35 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O35
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Crystal Structure Of The Kinase Domain Of Human C-Kit In Complex With A Type-Ii Inhibitor Bearing An Acrylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-05-27 Classification: SIGNALING PROTEIN Ligands: O2K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-27
Ligands: O2K
