Search Count: 11
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Cathepsin K Covalently Bound To A Cyano-Pyrimidine Inhibitor With Improved Selectivity Over Herg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: O47
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Cathepsin S In Complex With A Covalent Inhibitor With An Aldehyde Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O64, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O64, DMS
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Cathepsin K In Complex With A Covalent Inhibitor With A Ketoamide Warhead
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2010-12-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O96, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-22
Ligands: O96, SO4
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Cathepsin K Covalently Bound To A 2-Cyano Pyrimidine Inhibitor With A Benzyl P3 Group.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-10-06 Classification: HYDROLASE Ligands: SO4, O75 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: SO4, O75
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X-Ray Structure Of Cathepsin K Covalently Bound To A Triazine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: ORG, TFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ORG, TFA
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Cathepsin K In Complex With A Non-Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: SO4, KWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: SO4, KWZ
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Cathepsin K In Complex With A Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: KX1, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: KX1, SO4
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Crystal Structure Of An Alpha-L-Fucosidase Gh29 Trapped Covalent Intermediate From Bacteroides Thetaiotaomicron In Complex With 2- Fluoro-Fucosyl Fluoride Using An E288Q Mutant
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2010-02-02 Classification: HYDROLASE Ligands: FUF, SO4 |
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION
Release Date: 2010-02-02
Ligands: FUF, SO4
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Crystal Structure Of An Alpha-L-Fucosidase Gh29 From Bacteroides Thetaiotaomicron In Complex With A Novel Iminosugar Fucosidase Inhibitor
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-02-02 Classification: HYDROLASE Ligands: FHN, GOL, IMD |
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION
Release Date: 2010-02-02
Ligands: FHN, GOL, IMD
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Crystal Structure Of A Michaelis Complex Of Alpha-L-Fucosidase Gh29 From Bacteroides Thetaiotaomicron With The Synthetic Substrate 4- Nitrophenyl-Alpha-L-Fucose
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-02-02 Classification: HYDROLASE Ligands: SO4, JFZ |
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION
Release Date: 2010-02-02
Ligands: SO4, JFZ
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Crystal Structure Of An Alpha-L-Fucosidase Gh29 From Bacteroides Thetaiotaomicron
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2010-02-02 Classification: HYDROLASE Ligands: TRS, SO4, GOL |
Organism: Bacteroides thetaiotaomicron
Method: X-RAY DIFFRACTION
Release Date: 2010-02-02
Ligands: TRS, SO4, GOL
