Search Count: 38
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Arginase 2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2024-12-04 Classification: HYDROLASE Ligands: MN, A1H0B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: MN, A1H0B
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Arginase 2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2024-12-04 Classification: HYDROLASE Ligands: MN, A1H0A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: MN, A1H0A
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Arginase 2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-12-04 Classification: HYDROLASE Ligands: MN, DMS, PRO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: MN, DMS, PRO
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Arginase 2 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2024-11-27 Classification: HYDROLASE Ligands: MN, A1HZ9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-27
Ligands: MN, A1HZ9
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Crystal Structure Of Human Wdr5 In Complex With N-[(2'-Cyano[1,1'-Biphenyl]-4-Yl)Methyl]-3-Hydroxy-6-Methyl-4-Oxo-4H-Pyran-2-Carboxamide (Compound 1, Wdr5-Myc Ppi Inhibitor)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2023-06-28 Classification: ONCOPROTEIN/INHIBITOR Ligands: YJN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-28
Ligands: YJN
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Crystal Structure Of Human Wdr5 In Complex With (1M)-N-[(3,5-Difluoro[1,1'-Biphenyl]-4-Yl)Methyl]-6-Methyl-4-Oxo-1-(Pyridin-3-Yl)-1,4-Dihydropyridazine-3-Carboxamide (Compound 2, Wdr5-Myc Inhibitor)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2023-06-28 Classification: ONCOPROTEIN/INHIBITOR Ligands: YJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-28
Ligands: YJR
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Syk Kinase Domain In Complex With Macrocyclic Inhibitor 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2023-06-14 Classification: TRANSFERASE Ligands: QR7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: QR7
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 51A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 51A
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 52R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 52R
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: MG, L9W, 54N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: MG, L9W, 54N
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Eed In Complex With A Cyano-Benzofuran
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: CA, L9W, PV5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: CA, L9W, PV5
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Eed In Complex With A Triazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: L9W, GOL, EJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: L9W, GOL, EJR
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Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: LKT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: LKT, EDO
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Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: LKQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: LKQ
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Eed In Complex With A Triazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2019-09-25 Classification: PROTEIN BINDING Ligands: L9W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: L9W, GOL
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Eed In Complex With A Methyl-Thiazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-09-25 Classification: PROTEIN BINDING Ligands: CA, L9W, L9T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-25
Ligands: CA, L9W, L9T
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Novel Inhibitors Of Human Rhinovirus 3C Protease
Organism: Human rhinovirus 2
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-06-22 Classification: TRANSFERASE Ligands: GOL, PG4, PGE, HOV |
Organism: Human rhinovirus 2
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: GOL, PG4, PGE, HOV
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Novel Inhibitors Of Human Rhinovirus 3C Protease
Organism: Human rhinovirus 2
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-06-22 Classification: TRANSFERASE Ligands: 6OY |
Organism: Human rhinovirus 2
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6OY
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Human Jak1 Kinase In Complex With Compound 30 At 2.30 Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-11-25 Classification: TRANSFERASE Ligands: PEG, 5JG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: PEG, 5JG
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Tmk From S.Aureus In Complex With The Piperidinyl Thymine Class Inhibitor With A C5 Ethyl-Amine
Organism: Staphylococcus aureus (strain mu3 / atcc 700698)
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2015-02-11 Classification: TRANSFERASE Ligands: 43N |
Organism: Staphylococcus aureus (strain mu3 / atcc 700698)
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 43N
