Search Count: 43
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Crystal Structure Of Human Ldhb In Complex With Nadh, Oxamate, And Axko-0046
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-10-20 Classification: OXIDOREDUCTASE Ligands: NAI, OXM, EDO, H1U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-20
Ligands: NAI, OXM, EDO, H1U
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Crystal Structure Of Human Ldhb In Complex With Nadh
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-10-20 Classification: OXIDOREDUCTASE Ligands: NAI, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-20
Ligands: NAI, GOL
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P38 In Complex With T-3220137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-11-20 Classification: TRANSFERASE/INHIBITOR Ligands: MKP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: MKP
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Structure Of Rorgt In Complex With A Novel Inverse Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2019-07-17 Classification: nuclear protein/agonist Ligands: SO4, MPD, HQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: SO4, MPD, HQ7
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Structure Of Rorgt In Complex With A Novel Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-12 Classification: nuclear protein/agonist Ligands: EDO, HOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: EDO, HOJ
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping: Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-04-17 Classification: TRANSFERASE Ligands: J8S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J8S
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping - Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-04-17 Classification: TRANSFERASE/INHIBITOR Ligands: J9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J9G
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Structure Of Cdk12/Cyck In Complex With A Small Molecule Inhibitor N-(4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)-N-((1R,4R)-4-(Quinazolin-2-Ylamino)Cyclohexyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-08-29 Classification: TRANSFERASE/INHIBITOR Ligands: MG, 8M1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: MG, 8M1
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Structure Of Rorgt In Complex With A Novel Isoquinoline Inverse Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2018-03-21 Classification: transcription/agonist Ligands: MPD, E3S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: MPD, E3S
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Structure Of Rorgt In Complex With A Novel Inverse Agonist Tak-828.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-03-21 Classification: transcription/agonist Ligands: MPD, E3V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: MPD, E3V
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[1,2-B]Pyridazine-Based P38 Map Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-01-17 Classification: Transferase/Transferase Inhibitor Ligands: AQY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: AQY
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[1,2-B]Pyridazine-Based P38 Map Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: T75 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: T75
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Structure Of Rorgt In Complex With A Novel Inverse Agonist 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-01-03 Classification: SIGNALING PROTEIN Ligands: CFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-03
Ligands: CFG
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Design, Synthesis, And Evaluation Of The First Selective And Potent G-Protein-Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: QRW, SO4, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: QRW, SO4, MES
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Design, Synthesis, And Evaluation Of The First Selective And Potent G-Protein-Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-07-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 8PV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 8PV, SO4
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Crystal Structure Of Human Brr2 In Complex With T-3905516
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2017-07-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, 8LS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: GOL, 8LS
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Crystal Structure Of Human Brr2 In Complex With T-3935799
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2017-07-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: GOL, 8LP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: GOL, 8LP
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Crystal Structure Of Human Brr2 In Complex With T-1206548
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-07-19 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 8LV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-19
Ligands: 8LV
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The Crystal Structure Of Human S-Adenosylhomocysteine Hydrolase (Ahcy) Bound To Oxadiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-06-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAD, EDO, 9W1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: NAD, EDO, 9W1
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The Crystal Structure Of Human S-Adenosylhomocysteine Hydrolase (Ahcy) Bound To Benzothiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-06-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAD, 9W4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: NAD, 9W4, EDO