Search Count: 11
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Halk In Complex With Compound 7 N-((1S)-1-(5-Fluoropyridin-2-Yl)Ethyl)-1-(5-Methyl-1H-Pyrazol-3-Yl)-3-(Oxetan-3-Ylsulfonyl)-1H-Pyrrolo[2,3-B]Pyridin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-05-01 Classification: PROTEIN BINDING Ligands: HKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: HKJ
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Halk In Complex With Compound 9 (6-(((1S)-1-(5-Fluoropyridin-2-Yl)Ethyl)Amino)-1-(3-Methyl-1H-Pyrazol-5-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)(Morpholin-4-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2019-05-01 Classification: TRANSFERASE/INHIBITOR Ligands: J3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: J3Y
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Halk In Complex With Compound 1 (S)-N-(1-(2,4-Difluorophenyl)Ethyl)-3-(3-Methyl-1H-Pyrazol-5-Yl)Imidazo[1,2-B]Pyridazin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-05-01 Classification: TRANSFERASE/INHIBITOR Ligands: J4M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: J4M
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Egfr Kinase Domain Complexed With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-03-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W32, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: W32, SO4
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Egfr Kinase Domain Complexed With Compound 19B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W19, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: W19, SO4
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Egfr Kinase Domain T790M/L858R Mutant With Tak-285
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 03P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 03P
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Egfr Kinase Domain T790M/L858R Mutant With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W2P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: W2P
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Egfr Kinase Domain T790M/L858R Mutant With Hki-272
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: HKI, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: HKI, MES
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Egfr Kinase Domain T790M/L858R Mutant With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W2R, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: W2R, EDO
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Egfr Kinase Domain With Compound4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-01-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: W2R, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: W2R, SO4
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Her2 Kinase Domain Complexed With Tak-285
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.21 Å Release Date: 2011-11-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 03P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-11-23
Ligands: 03P
