Search Count: 205
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Apo Structure Of Pyr5 From Streptomyces Pyridomyceticus
Organism: Streptomyces pyridomyceticus
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2026-06-17 Classification: ISOMERASE Ligands: FLC |
Organism: Streptomyces pyridomyceticus
Method: X-RAY DIFFRACTION
Release Date: 2026-06-17
Ligands: FLC
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3-Bromopropiolate Treated Pyr5 From Streptomyces Pyridomyceticus
Organism: Streptomyces pyridomyceticus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-06-17 Classification: ISOMERASE |
Organism: Streptomyces pyridomyceticus
Method: X-RAY DIFFRACTION
Release Date: 2026-06-17
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Nicotinamide Riboside And Cd38: Covalent Inhibition And Live-Cell Labeling
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-11-06 Classification: HYDROLASE/INHIBITOR Ligands: NNR, RIB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: NNR, RIB
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X-Ray Structure Of Human Cd38 Catalytic Domain With 2'-Cl-Aranad+
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-06-03 Classification: HYDROLASE Ligands: ROJ, K, PO4, PEG, MPD, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-03
Ligands: ROJ, K, PO4, PEG, MPD, PGE
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A Structurally Dynamic N-Terminal Region Drives Function Of The Staphylococcal Peroxidase Inhibitor (Spin)
Organism: Homo sapiens, Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2017-12-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAG, BMA, CA |
Organism: Homo sapiens, Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: NAG, BMA, CA
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Novel 5-Azaindole Factor Viia Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2007-01-23 Classification: HYDROLASE/BLOOD CLOTTING Ligands: 7NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-23
Ligands: 7NH
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Discovery Of A Novel Hydroxy Pyrazole Based Factor Ixa Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2006-04-04 Classification: HYDROLASE/BLOOD CLOTTING Ligands: 6NH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-04-04
Ligands: 6NH
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Human Beta-Tryptase Ii With Inhibitor Cra-29382
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-03-21 Classification: HYDROLASE Ligands: C3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-21
Ligands: C3A
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Human Tryptase With 2-Amino Benzimidazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2006-03-07 Classification: HYDROLASE Ligands: AX7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-07
Ligands: AX7
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Human Beta Tryptase Ii With Inhibitor Cra-28427
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2006-03-07 Classification: HYDROLASE Ligands: C4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-03-07
Ligands: C4A
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Discovery Of Novel Heterocyclic Factor Viia Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2006-02-28 Classification: HYDROLASE/BLOOD CLOTTING Ligands: N1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-28
Ligands: N1H
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Factor Viia Inhibitors: Chemical Optimization, Preclinical Pharmacokinetics, Pharmacodynamics, And Efficacy In A Baboon Thrombosis Model
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2006-02-14 Classification: BLOOD CLOTTING Ligands: C1B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: C1B
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Human Beta-Tryptase Ii Complexed With 4-Piperidinebutyrate To Make Acylenzyme
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2006-02-14 Classification: HYDROLASE Ligands: C1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: C1R
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Bovine Trypsin Bound By 4-Piperidinebutyrate To Make Acylenzyme Complex
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2006-02-14 Classification: HYDROLASE Ligands: CA, C1R |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: CA, C1R
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Bovine Trypsin Complexed With 2-Aminobenzamidazole
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2006-02-14 Classification: HYDROLASE Ligands: CA, AX7 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2006-02-14
Ligands: CA, AX7
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Human Beta Tryptase Ii Complexed With Activated Ketone Inhibitor Cra-29382
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2006-02-09 Classification: HYDROLASE Ligands: C3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-02-09
Ligands: C3A
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Expression, Crystallization And Three-Dimensional Structure Of The Catalytic Domain Of Human Plasma Kallikrein: Implications For Structure-Based Design Of Protease Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2005-10-11 Classification: BLOOD CLOTTING, HYDROLASE Ligands: BEN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-11
Ligands: BEN
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Expression, Crystallization And The Three-Dimensional Structure Of The Catalytic Domain Of Human Plasma Kallikrein: Implications For Structure-Based Design Of Protease Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2005-10-11 Classification: BLOOD CLOTTING, HYDROLASE Ligands: PO4, BEN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-10-11
Ligands: PO4, BEN
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: 696, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: 696, CIT
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: ESI, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: ESI, CIT
