Search Count: 12
![]() |
Crystal Structure Of C-Met-D1228N In Complex With Kin-7615
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: A1AB1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: A1AB1
![]() |
The X-Ray Co-Crystal Structure Of Human Fgfr3 And Kin-3248
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2024-02-07 Classification: TRANSFERASE/INHIBITOR Ligands: MLT, WGF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: MLT, WGF
![]() |
The X-Ray Co-Crystal Structure Of Human Fgfr3 And Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2024-02-07 Classification: TRANSFERASE/INHIBITOR Ligands: CL, WIQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: CL, WIQ
![]() |
The X-Ray Co-Crystal Structure Of Human Fgfr3 V555M And Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2024-02-07 Classification: TRANSFERASE/INHIBITOR Ligands: SO4, WIQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: SO4, WIQ, EDO
![]() |
Crystal Structure Of Lysine Specific Demethylase 1 (Lsd1) With Cc-90011
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2020-10-21 Classification: FLAVOPROTEIN Ligands: V0Y, FAD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-21
Ligands: V0Y, FAD
![]() |
Crystal Structure Of Kdm4 With The Small Molecule Inhibitor Qc6352
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9DJ
![]() |
Crystal Structure Of Human Kdm4 With Small Molecule Inhibitor Qc5714
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-09-27 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: NI, ZN, 9FJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NI, ZN, 9FJ
![]() |
Fragment-Based Discovery Of A Small Molecule Reversible Inhibitor Of Bruton'S Tyrosine Kinase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-07-01 Classification: TRANSFERASE Ligands: IMD, IPA, EDO, 4L6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, EDO, 4L6
![]() |
Crystal Structure Of Bruton'S Tyrosine Kinase Bound To A Cinnoline Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-07-01 Classification: Transferase/Transferase Inhibitor Ligands: IMD, IPA, DMS, 4RU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, DMS, 4RU
![]() |
Crystal Structure Of Bruton'S Tyrosine Kinase In Complex With A Substituted Cinnoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-07-01 Classification: Transferase/Transferase Inhibitor Ligands: IMD, IPA, DMS, 4RV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-01
Ligands: IMD, IPA, DMS, 4RV
![]() |
Crystal Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek 1) In Complex With Ligand And Mgatp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2011-02-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ATP, MG, IZG, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-02-23
Ligands: ATP, MG, IZG, ACT
![]() |
Crystal Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek 1) In Complex With Ligand And Mgadp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-07-28 Classification: TRANSFERASE Ligands: ADP, MG, LSG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-07-28
Ligands: ADP, MG, LSG
