Search Count: 29
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Linked Kdm5A Jmj Domain Bound To The Inhibitor Gsk-J1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: K0I, MN, GOL, SO4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: K0I, MN, GOL, SO4, DMS
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Linked Kdm5A Jmj Domain Bound To The Inhibitor N43 I.E. 3-((6-(4-Acryloyl-1,4-Diazepan-1-Yl)-2-(Pyridin-2-Yl)Pyrimidin-4-Yl)Amino)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: H6G, MN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: H6G, MN
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Linked Kdm5A Jmj Domain Bound To The Inhibitor N44 I.E. 3-((2-(Pyridin-2-Yl)-6-(4-(Vinylsulfonyl)-1,4-Diazepan-1-Yl)Pyrimidin-4-Yl)Amino)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: H6J, MN, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: H6J, MN, GOL, DMS
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Linked Kdm5A Jmj Domain Bound To The Inhibitor N49 I.E. 2-((2-Chlorophenyl)(2-(1-Methylpyrrolidin-2-Yl)Ethoxy)Methyl)Thieno[3,2-B]Pyridine-7-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: H6S, H6T, MN, DMS, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: H6S, H6T, MN, DMS, SO4, EDO
 |
Linked Kdm5A Jmj Domain Bound To The Covalent Inhibitor N69 I.E. [2-((3-Acrylamidophenyl)(2-(Piperidin-1-Yl)Ethoxy)Methyl)Thieno[3,2-B]Pyridine-7-Carboxylic Acid]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: H74, MN, GOL, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: H74, MN, GOL, DMS, EDO
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Linked Kdm5A Jmj Domain Bound To Inhibitor N70 I.E.[2-((3-Aminophenyl)(2-(Piperidin-1-Yl)Ethoxy)Methyl)Thieno[3,2-B]Pyridine-7-Carboxylic Acid]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: H6V, MN, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: H6V, MN, GOL, EDO
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Linked Kdm5A Jmj Domain Forming Covalent Bond To Inhibitor N71 I.E. 2-((3-(4-(Dimethylamino)But-2-Enamido)Phenyl)(2-(Piperidin-1-Yl)Ethoxy)Methyl)Thieno[3,2-B]Pyridine-7-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2018-11-21 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: H77, HZV, HZM, MN, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-21
Ligands: H77, HZV, HZM, MN, GOL, DMS
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Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)(Propoxy)Methyl)-1H-Pyrrolo[3,2-B]Pyridine (Compound N9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DKP, MN, DMS, GOL, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DKP, MN, DMS, GOL, EDO, SO4
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)(2-(Piperidin-1-Yl)Ethoxy)Methyl)-1L2-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid (Compound N40)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DQG, MN, GOL, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DQG, MN, GOL, DMS, EDO
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)(2-(4,4-Difluoropiperidin-1-Yl)Ethoxy)Methyl)-1H-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid(Compound N41)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DKS, MN, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DKS, MN, GOL, DMS
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)((4,4-Difluorocyclohexyl)Methoxy)Methyl)-1H-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid(Compound N42)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DKV, MN, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DKV, MN, GOL, EDO
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)(2-(1-Methylpyrrolidin-2-Yl)Ethoxy)Methyl)-1H-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid(Compound 46)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DLJ, MN, EDO, DMS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DLJ, MN, EDO, DMS, GOL
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)(2-(1-Methyl-1H-Imidazol-2-Yl)Ethoxy)Methyl)-1H-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid (Compound N47)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE Ligands: DNV, MN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DNV, MN, GOL
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Linked Kdm5A Jmj Domain Bound To The Inhibitor (R)-2-((2-Chlorophenyl)(2-(Piperidin-1-Yl)Ethoxy)Methyl)-1L2-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid (Compound N51)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DO1, MN, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DO1, MN, DMS
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor (S)-2-((2-Chlorophenyl)(2-(Piperidin-1-Yl)Ethoxy)Methyl)-1L2-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid (Compound N52)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DQG, MN, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DQG, MN, DMS, EDO
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor (R)-N-(1-(3-Isopropyl-1H-Pyrazole-5-Carbonyl)Pyrrolidin-3-Yl)Cyclopropanecarboxamide (Compound N54)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: MN, GOL, 90V, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: MN, GOL, 90V, EDO
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Linked Kdm5A Jmj Domain Bound To The Inhibitor (S)-N-(1-(3-Isopropyl-1H-Pyrazole-5-Carbonyl)Pyrrolidin-3-Yl)Cyclopropanecarboxamide (Compound N55)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DQJ, MN, DMS, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DQJ, MN, DMS, GOL, EDO
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Linked Kdm5A Jmj Domain Bound To The Inhibitor 5-(1-(Tert-Butyl)-1H-Pyrazol-4-Yl)-6-Isopropyl-7-Oxo-4,7-Dihydropyrazolo[1,5-A]Pyrimidine-3-Carbonitrile (Compound N75/Cpi-48)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DQS, MN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DQS, MN, EDO, GOL
 |
Linked Kdm5A Jmj Domain Bound To The Inhibitor 2-((2-Chlorophenyl)(3-(Piperidin-1-Yl)Propoxy)Methyl)-1H-Pyrrolo[3,2-B]Pyridine-7-Carboxylic Acid (Compound N48)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-03-28 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: DNY, MN, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: DNY, MN, EDO, GOL
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Linked Kdm5A Jmj Domain Bound To The Inhibitor C49 (2-{[(2-{[(E)-2-(Dimethylamino)Ethenyl](Ethyl)Amino}-2-Oxoethyl)Amino]Methyl}Pyridine-4-Carboxylic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2016-07-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: MMK, MN, GOL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: MMK, MN, GOL, EDO