Search Count: 45,642
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R68, BU3 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R68, BU3
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R69 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R69
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R96 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R96
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R68 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R68
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R69, BU3 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R69, BU3
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R94 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R94
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Crystal Structures Of Protein Kinase B Selective Inhibitors In Complex With Protein Kinase A And Mutants
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2005-09-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R55 |
Organism: Bos taurus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2005-09-17
Ligands: R55
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The Catalytic Subunit Of Camp-Dependent Protein Kinase In Complex With Rho-Kinase Inhibitor H-1152P
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2003-12-16 Classification: Transferase/Transferase Inhibitor Ligands: H52, MG8 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-12-16
Ligands: H52, MG8
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The Catalytic Subunit Of Camp-Dependent Protein Kinase In Complex With Rho-Kinase Inhibitor Fasudil (Ha-1077)
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2003-12-16 Classification: Transferase/Transferase Inhibitor Ligands: M77 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-12-16
Ligands: M77
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The Catalytic Subunit Of Camp-Dependent Protein Kinase (Pka) In Complex With Rho-Kinase Inhibitor Y-27632
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2003-12-16 Classification: Transferase/Transferase Inhibitor Ligands: Y27 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-12-16
Ligands: Y27
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Nemo/Ikk Association Domain Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2008-04-22 Classification: Transferase/Transcription |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
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Co-Crystal Structure Of Lipid Kinase Pi3K Alpha With A Selective Phosphatidylinositol-3 Kinase Alpha Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-05-18 Classification: transferase/transferase inhibitor Ligands: 4Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 4Q2
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Co-Crystal Structures Of The Lipid Kinase Pi3K Alpha With Pan And Isoform Selective Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SCN, 1LT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: SCN, 1LT
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Crystal Structure Of The Complex Of Human Mitogen Activated Protein Kinase Kinase 5 Phox Domain (Map2K5-Phox) With Human Mitogen Activated Protein Kinase Kinase Kinase 2 Phox Domain (Map3K2-Phox)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2006-11-28 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
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Crystal Structure Of The Complex Of Human Mitogen Activated Protein Kinase Kinase 5 Phox Domain (Map2K5-Phox) With Human Mitogen Activated Protein Kinase Kinase Kinase 3 (Map3K3B-Phox)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2006-12-12 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-12
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Structure Of Camp-Dependent Protein Kinase Complexed With (4R,2S)-5'-(4-(4-Chlorobenzyloxy)Pyrrolidin-2-Ylmethanesulfonyl)Isoquinoline
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-11-02 Classification: TRANSFERASE/INHIBITOR Ligands: CQP |
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-02
Ligands: CQP
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Structure Of Camp-Dependent Protein Kinase Complexed With Isoquinoline-5-Sulfonic Acid (2-(2-(4-Chlorobenzyloxy)Ethylamino) Ethyl)Amide
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2005-11-02 Classification: TRANSFERASE/INHIBITOR Ligands: I5S |
Organism: Bos taurus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-11-02
Ligands: I5S
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Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: X3N, ZWE
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Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To H1047R Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERSE INHIBITOR Ligands: EDO, X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: EDO, X3N, ZWE
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Phospho-Erk2 Bound To Bivalent Inhibitor Sbp2
Organism: Homo sapiens, Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-07-26 Classification: TRANSFERASE/INHIBITOR Ligands: GOL, FRZ, 90A |
Organism: Homo sapiens, Hiv-1 m:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: GOL, FRZ, 90A
