Search Count: 8
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Crystal Structure Of Hpk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2YE
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Crystal Structure Of Hpk1 In Complex With Gne1858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F97, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: F97, EDO, MES
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Crystal Structure Of Hpk1 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2WI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2WI, SO4
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Crystal Structure Of Hpk1 In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2TR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2TR
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1.98A Structure Of Gsk945237 With S.Aureus Dna Gyrase And Singly Nicked Dna
Organism: Staphylococcus aureus, Staphylococcus aureus (strain n315), Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-05-25 Classification: ISOMERASE Ligands: MN, GOL, CL, 6EJ |
Organism: Staphylococcus aureus, Staphylococcus aureus (strain n315), Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, GOL, CL, 6EJ
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2.5A Structure Of Gsk945237 With S.Aureus Dna Gyrase And Dna.
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-05-25 Classification: ISOMERASE Ligands: MN, GOL, 6EJ |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, GOL, 6EJ
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Discovery Of Thiazolobenzoxepin Pi3-Kinase Inhibitors That Spare The Pi3-Kinase Beta Isoform
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-08-28 Classification: Transferase/Transferase Inhibitor Ligands: 1JV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-28
Ligands: 1JV
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Novel Hydroxyl Tricyclics (E.G. Gsk966587) As Potent Inhibitors Of Bacterial Type Iia Topoisomerases
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-08-07 Classification: ISOMERASE Ligands: MN, AE8 |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: MN, AE8
