Search Count: 46
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Crystal Structure Of Mastl Kinase Domain In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2025-01-22 Classification: TRANSFERASE/INHIBITOR Ligands: A1AAE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: A1AAE
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Crystal Structure Of Map4K4 In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2025-01-22 Classification: TRANSFERASE/INHIBITOR Ligands: A1AAA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: A1AAA
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1E
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: SO4, A1A1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: SO4, A1A1D
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1C
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1B, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1B, CL
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Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Compound 53
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2024-12-18 Classification: TRANSFERASE Ligands: A1A1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: A1A1A
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-[6-Chloro-4-(9-Methyl-1-Oxa-4,9-Diazaspiro[5.5]Undec-4-Yl)-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl]Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2023-04-05 Classification: TRANSFERASE Ligands: XXF, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF, SO4
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(3R,5S)-3-Amino-5-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(2S,5R)-5-Amino-2-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3O
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Pkceta Kinase Domain In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: XXF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF
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Pkceta Kinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
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Structure Of Human Anaplastic Lymphoma Kinase Domain In Complex With (4-[6-Amino-5-[(1~{R})-1-[5-Fluoro-2-(Triazol-2-Yl)Phenyl]Ethoxy]-3-Pyridyl]Isoindolin-1-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2022-06-29 Classification: TRANSFERASE Ligands: 25J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-29
Ligands: 25J
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Structure Of Human Anaplastic Lymphoma Kinase Domain In Complex With ((2~{R})-2-[5-[6-Amino-5-[(1~{R})-1-[5-Fluoro-2-(Triazol-2-Yl)Phenyl]Ethoxy]-3-Pyridyl]-4-Methyl-Thiazol-2-Yl]Propane-1,2-Diol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2022-06-29 Classification: TRANSFERASE Ligands: AWJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-29
Ligands: AWJ
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Crystal Structure Of Nonphosphorylated, Hpk1 Kinase Domain In Complex With Sunitinib In The Inactive State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Crystal Structure Of Diphosphorylated Hpk1 Kinase Domain In Complex With Sunitinib In The Active State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2019-05-01 Classification: SIGNALING PROTEIN Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Sunitinib In The Inactive State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Structure Of Human Anaplastic Lymphoma Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-02-20 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
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Structure Of The Axl Kinase Domain In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.84 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: 7YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 7YS
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Crystal Structure Of The Mer Kinase Domain In Complex With A Macrocyclic Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-07-26 Classification: Transferase/Transferase Inhibitor Ligands: 7YS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-26
Ligands: 7YS