Search Count: 24
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Crystal Structure Of Cdk2 Bound By Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1INI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1INI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 11 (Azd8421)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOP
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Induced Myeloid Leukemia Cell Differentiation Protein Fabcomplex In Complex With Compound 1
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2023-05-24 Classification: APOPTOSIS Ligands: VF8 |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: VF8
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Induced Myeloid Leukemia Cell Differentiation Protein Fabcomplex In Complex With Azd5991
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-12-26 Classification: APOPTOSIS Ligands: E4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4W
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Mcl1 In Complex With An Indole Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-12-26 Classification: IMMUNE SYSTEM Ligands: E4Q, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4Q, EDO
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Mcl1 In Complex With Indole Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-12-26 Classification: IMMUNE SYSTEM Ligands: E4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4K
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Human Pim1 Kinase In Complex With Compound 12B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2018-03-21 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: EDO, MVG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: EDO, MVG, SO4
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Crystal Structure Of Human Cdk12/Cyclink In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2017-12-27 Classification: TRANSFERASE/INHIBITOR Ligands: MG, CJM, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: MG, CJM, EDO
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Mcl1 Fab Complex In Complex With Compound 29
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2017-01-18 Classification: IMMUNE SYSTEM Ligands: 7LT |
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 7LT
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Mcl1 Fab Complex In Complex With Compound 21
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2017-01-18 Classification: IMMUNE SYSTEM Ligands: 7LW |
Organism: Mus musculus, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-18
Ligands: 7LW
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Crystal Structure Of Mcl1 With Compound 1
Organism: Mus musculus, homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-01-11 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Mus musculus, homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
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Tankyrase 1 With Phthalazinone 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-03-02 Classification: Transferase/Transferase Inhibitor Ligands: BU3, 5N8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: BU3, 5N8, ZN
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Tankyrase 1 With Phthalazinone 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-11-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, 5N2, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: EDO, 5N2, ZN, ACT
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Tankyrase In Complex With Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-05-13 Classification: TRANSFERASE/INHIBITOR Ligands: GOL, 3J1, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: GOL, 3J1, ZN
