Search Count: 15
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Crystal Structure Of 6-Fluoropyrazolo[1,5-A]Pyridine Derivative Bound To Kit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2026-08-05 Classification: TRANSFERASE Ligands: A1DJF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1DJF
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Crystal Structure Of Casdatifan Bound To Hif2A-B*:Arnt-B* Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2026-02-18 Classification: TRANSCRIPTION Ligands: A1I0H, FMT, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: A1I0H, FMT, MG
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Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.96 Å Release Date: 2021-11-03 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V84 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-03
Ligands: V84
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Crystal Structure Of Human Pi3K-Gamma In Complex With Inhibitor Ipi-549
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V7Y, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V7Y, SO4
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Crystal Structure Of Human Pi3K-Gamma In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-09-16 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: V81, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: V81, SO4
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative Ab680 (Compound 55 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-09-16 Classification: HYDROLASE Ligands: ZN, CA, QDH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-16
Ligands: ZN, CA, QDH
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With Aopcp Derivative A830 (Compound 16 In Publication) In The Closed Form (Crystal Form Iii)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-07-22 Classification: HYDROLASE Ligands: ZN, CA, QCQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ZN, CA, QCQ
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2396 (Compound 74 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1H
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A2410 (Compound 53 In Publication) In The Closed Form In Crystal Form Iv
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, PO4, O1Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, PO4, O1Q
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Human Ecto-5'-Nucleotidase (Cd73) In Complex With A1618 (Compound 1B In Publication) In The Closed State In Crystal Form Iii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-04-22 Classification: HYDROLASE Ligands: ZN, CA, O1T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
Ligands: ZN, CA, O1T
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Hiv Integrase Catalytic Domain Containing F185K Mutation Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Hiv Integrase Catalytic Domain Containing F185K + A124T Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Hiv Integrase Catalytic Domain Containing F185K + A124N + T125S Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Hiv Integrase Catalytic Domain Containing F185K + A124N + T125A Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Crystal Structure Of The Hiv-1 Integrase Catalytic Domain With Gsk1264
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-06-11 Classification: VIRAL PROTEIN Ligands: 2SQ, CAC, SO4 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 2SQ, CAC, SO4
