Search Count: 10
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Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2024-08-14 Classification: CELL CYCLE Ligands: GTP, MG, GDP, UIY, SO4 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-04-13 Classification: TRANSFERASE Ligands: CL, EKR |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-04-13 Classification: TRANSFERASE Ligands: CL, EKF |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-04-13 Classification: TRANSFERASE Ligands: CL, EJR |
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In Vitro And In Vivo Characterization Of A Novel, Highly Potent P53-Mdm2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-09-26 Classification: CELL CYCLE Ligands: EYH, CL |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2018-08-22 Classification: LIGASE Ligands: 9QW, CL |
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Discovery Of A Novel Class Of Highly Potent Inhibitors Of The P53-Mdm2 Interaction By Structure-Based Design Starting From A Conformational Argument
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2016-09-07 Classification: CELL CYCLE Ligands: 6ZT, SO4, CL |
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Discovery Of Nvp-Cgm097 - A Highly Potent And Selective Mdm2 Inhibitor Undergoing Phase 1 Clinical Trials In P53Wt Tumors: Hdm2 (Mdm2) Complexed With Nvp-Cgm097
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-07-29 Classification: CELL CYCLE Ligands: 4T4, CL |
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Discovery Of Nvp-Cgm097 - A Highly Potent And Selective Mdm2 Inhibitor Undergoing Phase 1 Clinical Trials In P53Wt Tumors: Hdm2 (Mdm2) Complexed With Cpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2015-07-29 Classification: CELL CYCLE Ligands: 4TH, CL |
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Discovery Of Dihydroisoquinolinone Derivatives As Novel Inhibitors Of The P53-Mdm2 Interaction With A Distinct Binding Mode: Hdm2 (Mdm2) Complexed With Cpd5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-07-22 Classification: LIGASE Ligands: 4SS, SO4 |










