Search Count: 18
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Structure-Activity Relationship Studies Of Allosteric Inhibitors Of Eya2 Tyrosine Phosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.49 Å Release Date: 2021-12-29 Classification: TRANSCRIPTION Ligands: 1RI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-29
Ligands: 1RI
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Structure-Activity Relationship Studies Of Allosteric Inhibitors Of Eya2 Tyrosine Phosphatase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2021-12-29 Classification: TRANSCRIPTION Ligands: 1SI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-29
Ligands: 1SI
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Crystal Structure Of Wild Type Mnk2 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2020-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BV9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: BV9
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Crystal Structure Of Pkciota In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.26 Å Release Date: 2019-06-26 Classification: TRANSFERASE Ligands: AFU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: AFU
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Structural Basis For An Allosteric Eya2 Phosphatase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2019-06-05 Classification: TRANSCRIPTION Ligands: 9FX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: 9FX
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Crystal Structure Of Smyd3 In Complex With Covalent Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2018-08-08 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 8HF, SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: ZN, 8HF, SAM
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Crystal Structure Of Zika Virus Ns3 Protease In Complex With A Small Molecule Inhibitor
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-03-21 Classification: VIRAL PROTEIN/INHIBITOR Ligands: BEZ |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: BEZ
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Crystal Structure Of Zika Virus Ns3 Protease In Complex With A Dipeptide Inhibitor
Organism: Zika virus
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2018-03-21 Classification: VIRAL PROTEIN/INHIBITOR Ligands: 7HS |
Organism: Zika virus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: 7HS
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Tankyrase In Complex With 2-Hydroxy-4-Methylquinoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-07-10 Classification: TRANSFERASE Ligands: AJ2, ZN, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: AJ2, ZN, SO4
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Tankyrase 2 In Complex With 4-Chloro-1,2-Dihydrophatalzin-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-07-10 Classification: TRANSFERASE Ligands: ZN, SO4, 495 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: ZN, SO4, 495
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Tankyrase In Complex With 7-(2-Fluorophenyl)-4-Methyl-1,2-Dihydroquinolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2013-06-26 Classification: TRANSFERASE Ligands: ZN, SO4, AJ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: ZN, SO4, AJ4
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Tankyrase 2 In Complex With 7-(4-Amino-2-Chlorophenyl)-4-Methylquinolin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2013-06-26 Classification: TRANSFERASE Ligands: ZN, SO4, AJ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: ZN, SO4, AJ6
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Tankyrase 2 In Complex With 3-Chloro-4-(4-Methyl-2-Oxo-1,2-Dihydroquinolin-7-Yl)-N-[2-(Morpholin-4-Yl)Ethyl]Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2013-06-26 Classification: TRANSFERASE Ligands: ZN, SO4, AJ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: ZN, SO4, AJ7
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Tankyrase 2 In Complex With 3-Chloro-N-(2-Methoxyethyl)-4-(4-Methyl-2-Oxo-1,2-Dihydroquinolin-7-Yl)Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2013-06-26 Classification: TRANSFERASE Ligands: ZN, SO4, AJ5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: ZN, SO4, AJ5
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Tankyrase 2 In Complex With 3-Chloro-4-(4-Methyl-2-Oxo-1,2-Dihydroquinolin-7-Yl)Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-06-26 Classification: TRANSFERASE Ligands: ZN, SO4, AJ8, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-06-26
Ligands: ZN, SO4, AJ8, GOL
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Crystal Structure Of Wild Type Human Lipocalin Pgds Bound With Peg Mme 2000
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2013-03-20 Classification: ISOMERASE Ligands: 1PG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: 1PG
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Crystal Structure Of Wild Type Human Lipocalin Pgds In Complex With Substrate Analog U44069
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2013-03-20 Classification: ISOMERASE Ligands: PWZ, SCN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: PWZ, SCN
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Crystal Structure Of The Human Lipocalin-Type Prostaglandin D Synthase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-01-12 Classification: ISOMERASE Ligands: CL, SCN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: CL, SCN
