Search Count: 14
![]() |
Khk Bound To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1C0G, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1C0G, SO4
![]() |
Khk Bound To Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1C0I, FRU, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1C0I, FRU, SO4, GOL
![]() |
Khk Bound To Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1C0K, FRU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1C0K, FRU, SO4
![]() |
Khk Bound To Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1C0J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1C0J, SO4
![]() |
Khk Bound To Gs-1291269
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2026-01-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1C0H, FRU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-07
Ligands: A1C0H, FRU
![]() |
Hiv-1 Reverse Transcriptase In Complex With 5-Membered Bicyclic Core Nnrti
Organism: Hiv whole-genome vector aa1305#18
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2023-02-01 Classification: VIRAL PROTEIN Ligands: YO9, TLA |
Organism: Hiv whole-genome vector aa1305#18
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: YO9, TLA
![]() |
Hiv-1 Reverse Transcriptase In Complex With 6-Membered Bicyclic Core Nnrti
Organism: Hiv whole-genome vector aa1305#18
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2023-02-01 Classification: VIRAL PROTEIN Ligands: ZJ2, TLA |
Organism: Hiv whole-genome vector aa1305#18
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: ZJ2, TLA
![]() |
Hiv-1 Reverse Transcriptase In Complex With 7-Membered Bicyclic Core Nnrti
Organism: Hiv whole-genome vector aa1305#18
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2023-02-01 Classification: VIRAL PROTEIN Ligands: XRL, TLA |
Organism: Hiv whole-genome vector aa1305#18
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: XRL, TLA
![]() |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 3) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 7HG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 7HG
![]() |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 5) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78E
![]() |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 6) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78R
![]() |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 7) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78X
![]() |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 8) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 838, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 838, SO4
![]() |
Hiv-1 Reverse Transcriptase In Complex With A 2,6-Difluorophenyl Dapy Analog
Organism: Human immunodeficiency virus type 1 group m subtype b (isolate hxb2), Human immunodeficiency virus type 1 group m subtype b (isolate lw123)
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-06-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: IB1 |

