Search Count: 8
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Discovery Of Mta-Cooperative Prmt5 Inhibitors From Co-Factor Directed Dna-Encoded Library Screens
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2025-05-07 Classification: TRANSFERASE/INHIBITOR Ligands: A1B6Y, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-07
Ligands: A1B6Y, MTA
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From Dna-Encoded Library Screening To Am-9747 - An Mta-Cooperative Prmt5 Inhibitor With Potent Oral In Vivo Efficacy
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-03-26 Classification: TRANSFERASE/INHIBITOR Ligands: A1BQW, MTA, GOL, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-26
Ligands: A1BQW, MTA, GOL, PEG, DMS
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14-3-3 Sigma In Complex With Foxo1 Pt24 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-07-31 Classification: PEPTIDE BINDING PROTEIN Ligands: B3P, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: B3P, GOL
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14-3-3 Sigma In Complex With Foxo1 Ps256 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-07-31 Classification: PEPTIDE BINDING PROTEIN Ligands: GOL, B3P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-31
Ligands: GOL, B3P
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Human Fxia In Complex With Small Molecule Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2016-01-20 Classification: HYDROLASE Ligands: GOL, J1J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: GOL, J1J, SO4
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Human Fxia In Complex With Small Molecule Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2016-01-20 Classification: HYDROLASE Ligands: GOL, IXA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: GOL, IXA, SO4
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Human Fxia In Complex With Small Molecule Inhibitors.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2016-01-20 Classification: HYDROLASE Ligands: GOL, E6U, SO4, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-20
Ligands: GOL, E6U, SO4, TRS
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Structural And Energetic Determinants For Hyperstable Variants Of Gb1 Obtained From In-Vitro Evolution
Organism: Streptococcus sp. 'group g'
Method: X-RAY DIFFRACTION Resolution:0.88 Å Release Date: 2009-08-18 Classification: PROTEIN BINDING Ligands: CA |
Organism: Streptococcus sp. 'group g'
Method: X-RAY DIFFRACTION
Release Date: 2009-08-18
Ligands: CA
