Search Count: 18
 |
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, NAG, A1JCF, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, NAG, A1JCF, PO4
 |
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, NAG, A1JCG, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, NAG, A1JCG, PO4
 |
Human Cd73 (Ecto 5'-Nucleotidase) In Complex With Compound 6 (Oric-533)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: ZN, CA, A1JCH, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: ZN, CA, A1JCH, PO4
 |
Egfr Exon20 Insertion Mutant Asv Bound With (S)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN,TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1IMS, CL, EDO, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1IMS, CL, EDO, GOL, PEG
 |
Egfr Exon20 Insertion Mutant Svd Bound With (S)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN,TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1IMS, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1IMS, EDO, GOL
 |
Egfr Exon20 Insertion Mutant Svd Bound With Stx-721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN,TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1A4E, CL, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1A4E, CL, EDO, GOL
 |
Wildtype Egfr Bound With (R)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.12 Å Release Date: 2025-05-14 Classification: ONCOPROTEIN Ligands: A1ILZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1ILZ
 |
Egfr Exon20 Insertion Mutant Npg Bound With (S)-3-((3-Chloro-2-Methoxyphenyl)Amino)-2-(3-((Tetrahydrofuran-2-Yl)Methoxy)Pyridin-4-Yl)-1,5,6,7-Tetrahydro-4H-Pyrrolo[3,2-C]Pyridin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2025-05-14 Classification: TRANSFERASE Ligands: A1IMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1IMS
 |
Egfr Exon20 Insertion Mutant Npg Bound With Stx-721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-05-14 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
 |
Wild-Type Egfr Bound With Stx-721
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2025-05-14 Classification: TRANSFERASE Ligands: CL, A1IMT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: CL, A1IMT
 |
Egfr Exon20 Insertion Mutant Npg Bound With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2025-01-29 Classification: TRANSFERASE Ligands: A1IEZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: A1IEZ
 |
Egfr Exon20 Insertion Mutant Npg Bound With Compound 39
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2025-01-29 Classification: TRANSFERASE Ligands: EDO, A1IE0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: EDO, A1IE0
 |
Wildtype Egfr Bound With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2025-01-29 Classification: ONCOPROTEIN Ligands: DTT, A1IEZ, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-29
Ligands: DTT, A1IEZ, CL
 |
Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: X3N, ZWE
 |
Stx-478, A Mutant-Selective, Allosteric Inhibitor Bound To H1047R Pi3Kalpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2023-09-06 Classification: TRANSFERASE/TRANSFERSE INHIBITOR Ligands: EDO, X3N, ZWE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-09-06
Ligands: EDO, X3N, ZWE
 |
Glucocorticoid Receptor In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2018-10-03 Classification: TRANSCRIPTION Ligands: HJ4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-03
Ligands: HJ4
 |
Pqr309 - A Potent, Brain-Penetrant, Orally Bioavailable, Pan-Class I Pi3K/Mtor Inhibitor As Clinical Candidate In Oncology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: A3W, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: A3W, SO4
 |
Structure Of Histone Lysine Demethylase Kdm5A In Complex With Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Inhibitor Ligands: NI, ZN, 50P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NI, ZN, 50P