Search Count: 10
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Human Idh1 R132C Mutant Complexed With Compound A.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-10-30 Classification: OXIDOREDUCTASE Ligands: AOU, NDP, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: AOU, NDP, CIT, GOL
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Crystal Structure Of Rip1 Kinase Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-21 Classification: Transferase/Transferase Inhibitor Ligands: EJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: EJY
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Structure Based Design Of Rip1 Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2018-03-21 Classification: Transferase/Transferase Inhibitor Ligands: EJP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: EJP
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Human Squalene Synthase In Complex With 2-(1-{2-[(4R,6S)-8-Chloro-6-(2,3-Dimethoxyphenyl)-4H,6H-Pyrrolo[1,2-A][4,1]Benzoxazepin-4-Yl]Acetyl}-4-Piperidinyl)Acetic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-12-19 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, D3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-12-19
Ligands: PO4, D3A
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Human Squalene Synthase In Complex With 1-{4-[{4-Chloro-2-[(2-Chlorophenyl)(Hydroxy)Methyl]Phenyl}(2,2-Dimethylpropyl)Amino]-4-Oxobutanoyl}Piperidine-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, D99 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: PO4, D99
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Human Squalene Synthase In Complex With N-[(3R,5S)-7-Chloro-5-(2,3-Dimethoxyphenyl)-1-Neopentyl-2-Oxo-1,2,3,5-Tetrahydro-4,1-Benzoxazepine-3-Acetyl]-L-Aspartic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: PO4, D9A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: PO4, D9A
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Human Squalene Synthase In Complex With (2R,3R)-2-Carboxymethoxy-3-[5-(2-Naphthalenyl)Pentyl]Aminocarbonyl-3-[5-(2-Naphthalenyl)Pentyloxy]Propionic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, D61, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-21
Ligands: MG, D61, PO4
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Gsk3Beta Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: G3B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: G3B
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X-Ray Co-Crystal Structure Of Glycogen Synthase Kinase 3Beta In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2009-03-10 Classification: TRANSFERASE Ligands: 34O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: 34O
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Glycogen Synthase Kinase 3Beta Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-03-10 Classification: TRANSFERASE Ligands: 3HT, 2HT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-10
Ligands: 3HT, 2HT
