Search Count: 37
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Crystal Structure Of Pim1 In Complex With A Pyrrolo-Pyrazinone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-10-05 Classification: TRANSFERASE Ligands: JYO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-05
Ligands: JYO
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Crystal Structure Of Human Choline Alpha In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-10-13 Classification: TRANSFERASE Ligands: U6T, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: U6T, EPE
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Crystal Structure Of Human Choline Alpha In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-10-13 Classification: TRANSFERASE Ligands: EPE, U6E, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: EPE, U6E, MG
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Crystal Structure Of Human Choline Alpha In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-10-13 Classification: TRANSFERASE Ligands: U6H, MG, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: U6H, MG, EPE
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The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7W |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: H7W
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The Catalytic Fragment Of Poly(Adp-Ribose) Polymerase Complexed With An Isoindolinone Inhibitor
Organism: Gallus gallus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: H7Z |
Organism: Gallus gallus
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: H7Z
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Crystal Structure Of The Alk Kinase Domain In Complex With Entrectinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: YMX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: YMX
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Crystal Structure Of The Alk Kinase Domain In Complex With Cmpd 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-04-06 Classification: TRANSFERASE Ligands: U4W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: U4W, GOL
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Structure Of Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: FSU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: FSU
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Structure Of Human Parp2 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: D7N
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Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: SO4, GOL, FSU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: SO4, GOL, FSU
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Structure Of Human Parp1 Catalytic Domain Bound To An Isoindolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2015-08-12 Classification: TRANSFERASE Ligands: D7N, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: D7N, SO4
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Novel Pyrrole Carboxamide Inhibitors Of Jak2 As Potential Treatment Of Myeloproliferative Disorders
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-04-29 Classification: TRANSFERASE Ligands: QUP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-29
Ligands: QUP
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B-Raf Kinase V600E Mutant In Complex With A Diarylthiazole B-Raf Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-12-10 Classification: TRANSFERASE Ligands: CQE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: CQE
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: GOL, VVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: GOL, VVQ
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: 953, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: 953, GOL
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Pyrrole-3-Carboxamides As Potent And Selective Jak2 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2014-07-23 Classification: TRANSFERASE Ligands: BJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-23
Ligands: BJG
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Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: H05 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: H05
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Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: 6LV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: 6LV
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Human Hsp90 Alpha N-Terminal Domain In Complex With An Aminotriazoloquinazoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2014-07-09 Classification: CHAPERONE Ligands: T62 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-09
Ligands: T62
