Search Count: 22
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Crystal Structure Of Fgfr2 Kinase Domain Gatekeeper Mutant V564F In Complex With Covalent Compound 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2021-02-10 Classification: SIGNALING PROTEIN Ligands: WFD, FLC, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: WFD, FLC, NA
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Crystal Structure Of Fgfr2 Kinase Domain Gatekeeper Mutant V564F In Complex With Covalent Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2021-02-10 Classification: SIGNALING PROTEIN Ligands: WF7, FLC, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: WF7, FLC, GOL
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Cps1 Bound To Allosteric Inhibitor H3B-374
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2021-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 374, ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: 374, ZN, EDO
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Cps1 Bound To Allosteric Inhibitor H3B-193
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-03-18 Classification: LIGASE/LIGASE INHIBITOR Ligands: ZN, Q5A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-18
Ligands: ZN, Q5A
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Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: SO4, D4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: SO4, D4Q
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Chk1 Kinase In Complex With Compound 44
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: D58, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D58, SO4
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Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: D4Z, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D4Z, SO4
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Crystal Structure Of Usp7 In Complex With The Non-Covalent Inhibitor, Ft671
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2017-10-18 Classification: HYDROLASE Ligands: 8WK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8WK
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Crystal Structure Of Usp7 In Complex With The Covalent Inhibitor, Ft827
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-10-18 Classification: HYDROLASE Ligands: 8WN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 8WN, EDO
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Tankyrase 1 With Phthalazinone 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2016-03-02 Classification: Transferase/Transferase Inhibitor Ligands: BU3, 5N8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-02
Ligands: BU3, 5N8, ZN
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Tankyrase 1 With Phthalazinone 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-11-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, 5N2, ZN, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: EDO, 5N2, ZN, ACT
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Tankyrase In Complex With Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-05-13 Classification: TRANSFERASE/INHIBITOR Ligands: GOL, 3J1, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: GOL, 3J1, ZN
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Human Tankyrase 1 With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2015-05-13 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, 3J5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-13
Ligands: ZN, 3J5
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Inhibitors Of Jak2 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2014-01-08 Classification: TRANSFERASE Ligands: LMM, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-08
Ligands: LMM, ACT
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Inhibitors Of Jak2 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2014-01-08 Classification: TRANSFERASE Ligands: XWW, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-08
Ligands: XWW, ACT
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Inhibitors Of Jak2 Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2013-04-17 Classification: TRANSFERASE Ligands: F9J, ACE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-17
Ligands: F9J, ACE
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Human Trka In Complex With The Inhibitor Az-23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2012-08-15 Classification: TRANSFERASE Ligands: V4Z, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: V4Z, ZN
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, YDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, YDI
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, GOL, YDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, GOL, YDK
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2012-01-25 Classification: TRANSFERASE Ligands: YDJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: YDJ, PO4