Search Count: 25
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Structure Of Cdk12/Cyck In Complex With A Small Molecule Inhibitor N-(4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)-N-((1R,4R)-4-(Quinazolin-2-Ylamino)Cyclohexyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2018-08-29 Classification: TRANSFERASE/INHIBITOR Ligands: MG, 8M1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-29
Ligands: MG, 8M1
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Optimization Of 3,5-Disubstitued Piperidine: Discovery Of Non-Peptide Mimetics As An Orally Active Renin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 7EK, PGE, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 7EK, PGE, PEG, DMS
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Optimization Of 3,5-Disubstitued Piperidine: Discovery Of Non-Peptide Mimetics As An Orally Active Renin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 7EJ, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: NAG, 7EJ, DMS, PEG
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2017-08-16 Classification: Transcription/Inhibitor Ligands: 80R, EDO, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 80R, EDO, K
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2017-08-16 Classification: Transcription/Inhibitor Ligands: 80L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 80L
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2017-07-05 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VU, PGE, PEG, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-05
Ligands: NAG, 6VU, PGE, PEG, DMS
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7ZF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7ZF
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7ZL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7ZL, EDO
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: YAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: YAM
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7ZO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7ZO
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-05-24 Classification: Transcription/Inhibitor Ligands: 7Z6, EDO, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-24
Ligands: 7Z6, EDO, K
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Coactivator-Associated Arginine Methyltransferase 1 With Tp-064
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-12-21 Classification: TRANSFERASE Ligands: SAH, 7VM, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-21
Ligands: SAH, 7VM, UNX
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Crystal Structure Of The Bcl6 Btb Domain In Complex With F1324
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-12-07 Classification: Transcription/Inhibitor Ligands: SO4 |
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: SO4
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Crystal Structure Of The Bcl6 Btb Domain In Complex With F1324(10-13)
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-12-07 Classification: Transcription/Inhibitor Ligands: EDO |
Organism: Homo sapiens, Enterobacteria phage t7
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: EDO
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2016-11-16 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VS, DMS, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-16
Ligands: NAG, 6VS, DMS, PEG
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Discovery Of Tak-272: A Novel, Potent And Orally Active Renin In-Hibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6VR, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 6VR, PEG
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 74U, PEG, NAG, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 74U, PEG, NAG, PGE
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 74V, PGE, DMS, 1PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 74V, PGE, DMS, 1PE
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 74Z, DMS, PEG, 1PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 74Z, DMS, PEG, 1PE
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Structure-Based Design Of A New Series Of N-Piperidin-3-Ylpyrimidine-5-Carboxamides As Renin Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-11-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, 74Y, PEG, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: NAG, 74Y, PEG, PGE