Search Count: 19
 |
Crystal Structure Of Irak4-Hsa Complexed With N-[(2R)-2-Fluoro-3-Hydroxy-3-Methylbutyl]-6-[(5-Fluoropyri-Yl)Amino]-4-[(Propan-2-Yl)Amino]Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2025-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZVD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: ZVD, SO4
 |
Crystal Structure Of Irak4-Hsa Complexed With Bms-986126; 6-((5-Cyano-2-Pyrimidinyl)Amino)-N-((2R)-2-Fluoro-3-Hydroxhylbutyl)-4-(Isopropylamino)Nicotinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2025-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZVG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: ZVG, SO4
 |
Crystal Structure Of Irak4-Hsa Complexed With Bms-986147; 6-{5-Cyano-1H-Pyrazolo[3,4-B]Pyridin-1-Yl}-N-[(2R)-2-Fluorroxy-3-Methylbutyl]-4-[(Propan-2-Yl)Amino]Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.76 Å Release Date: 2025-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, ZVA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: SO4, ZVA
 |
The Jak3 Kinase Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9Z4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: 9Z4
 |
Crystal Structure Of Pi3K Delta In Complex With A Trifluoro-Ethyl-Pyrazol-Pyrolotriazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: 9EM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: 9EM
 |
Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 9J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 9J4
 |
Structure Of Human Pregnane X Receptor Ligand Binding Domain With Adnectin-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-02-11 Classification: IMMUNE SYSTEM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
 |
Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound With Adnectin-1 And Compound-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2015-02-04 Classification: TRANSCRIPTION Ligands: 40U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 40U
 |
Structure Of Human Pregnane X Receptor Ligand Binding Domain With Compound-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-01-28 Classification: TRANSCRIPTION Ligands: GOL, 40U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: GOL, 40U
 |
Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2014-12-24 Classification: TRANSFERASE/INHIBITOR Ligands: 3QX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3QX
 |
Crystal Structure Of The Human Pxr-Lbd In Complex With N-{(2R)-1-[(4S)-4-(4-Chlorophenyl)-4-Hydroxy-3,3-Dimethylpiperidin-1-Yl]-3-Methyl-1-Oxobutan-2-Yl}-3-Hydroxy-3-Methylbutanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-08-27 Classification: TRANSCRIPTION/TRANSCRIPTION inhibitor Ligands: 2Q4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-08-27
Ligands: 2Q4, GOL
 |
P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-10-13 Classification: TRANSFERASE Ligands: 38P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 38P
 |
P38 Alpha Map Kinase Complexed With Pyrrolotriazine Inhibitor 7V
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2010-10-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 39P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-13
Ligands: 39P
 |
P38 Alpha Kinase Complexed With A 2-Aminothiazol-5-Yl-Pyrimidine Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2010-09-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3NW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: 3NW
 |
Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2008-04-15 Classification: TRANSFERASE Ligands: P39 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: P39
 |
P38 Alpha Map Kinase Complexed With Bms-640994
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-15 Classification: SIGNALING PROTEIN, TRANSFERASE Ligands: 304 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-15
Ligands: 304
 |
Morpholino Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-04-08 Classification: TRANSFERASE Ligands: P38 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: P38
 |
Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 279 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 279
 |
Phenylalanine Pyrrolotriazine P38 Alpha Map Kinase Inhibitor Compound 11J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: 287 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: 287