Search Count: 27
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Structure Of Eif2B Bound To A Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2026-06-03 Classification: SUGAR BINDING PROTEIN Ligands: SO4, A1DBY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: SO4, A1DBY
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Crystal Structure Of Wrn In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2025-06-18 Classification: HYDROLASE Ligands: A1CA4, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1CA4, ZN
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Crystal Structure Of Wrn In Complex With Compound 43
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-06-18 Classification: HYDROLASE Ligands: A1CA5, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1CA5, ZN
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Degrader-Induced Complex Between Ptpn2 And Crbn-Ddb1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2024-09-11 Classification: HYDROLASE Ligands: WO8, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2024-09-11
Ligands: WO8, ZN
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Crystal Structure Of Ptpn2 With A Protac
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2024-09-04 Classification: HYDROLASE Ligands: UB0, ACT, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: UB0, ACT, NA
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Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
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Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
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Crystal Structure Of Human Ptpn2 With Inhibitor Abbv-Cls-484
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2023-07-26 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: M5R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: M5R
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Brd4_Bd2-A-35165
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2017-06-28 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 89J
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Brd4_Bd2_A-1107604
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 0S6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 0S6
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Brd2 Bromodomain2 With A-1360579
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 87D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 87D
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Brd4_Bd2_A-1497627
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 89D
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Brd4_Bd2_A-1412838
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 88M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 88M
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Brd4_Bd2_A-1342843
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2017-05-10 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: 89G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-10
Ligands: 89G
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Crystal Structure Of Hsetd8 In Complex With Histone H4K20 Norleucine Mutant Peptide And S-Adenosylmethionine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2016-12-07 Classification: TRANSFERASE Ligands: SAM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-12-07
Ligands: SAM
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Selective Aminopyridine-Based C-Jun N-Terminal Kinase Inhibitors With Cellular Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2006-06-06 Classification: TRANSCRIPTION Ligands: SO4, 877 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-06-06
Ligands: SO4, 877
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Ptp1B Complexed With Isoxazole Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2004-10-19 Classification: HYDROLASE Ligands: IX1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-10-19
Ligands: IX1
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Monoacid-Based, Cell Permeable, Selective Inhibitors Of Protein Tyrosine Phosphatase 1B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2003-10-28 Classification: HYDROLASE Ligands: 429 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-10-28
Ligands: 429
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Dual-Site Potent, Selective Protein Tyrosine Phosphatase 1B Inhibitor Using A Linked Fragment Strategy And A Malonate Head On The First Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2003-09-16 Classification: HYDROLASE Ligands: 941 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-16
Ligands: 941
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A Highly Efficient Approach To A Selective And Cell Active Ptp1B Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2003-09-16 Classification: HYDROLASE Ligands: 234 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2003-09-16
Ligands: 234
